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4-({[(4-fluorophenyl)methyl](1-hydroxybutan-2-yl)amino}methyl)benzonitrile
(3S,4R)-4-(2-methoxyphenyl)-1-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)pyrrolidine-3-carboxylic acid
methyl (2S)-1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
1-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-1,4-diazepan-5-one
1-[4-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)phenyl]-1H-pyrazole
N-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzoic acid
(propan-2-yl)({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-benzotriazole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
N,N-diethyl-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazol-5-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-3-ol
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
7-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-[(3,5-difluorophenyl)methyl]-8-(thiophen-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 4-{[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]carbamoyl}butanoate
5-{1-[2-(4-chlorophenyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]acetamide
3-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-(dimethyl-1,2-oxazol-4-yl)benzamide
(2S,4S)-4-[(adamantan-2-yl)amino]-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-(furan-2-carbonyl)-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-amine
1-(cyclopentylmethyl)-3-(4-fluorophenoxy)azetidine
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(oxolan-3-yl)acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-4-carboxamide
4-(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1H-imidazol-5-yl)-2,1,3-benzoxadiazole
N-cyclobutyl-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
5,6-dimethyl-2-(4-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-(3-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
N-ethyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-({[(3-chlorophenyl)carbamoyl]amino}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{2-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[(2S)-butan-2-yl]-2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide
3-[5-(cyclopropylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
7-(2-hydroxyethyl)-2-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-cyclopentanecarbonyl-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
9-[5-(hydroxymethyl)furan-2-carbonyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-4-(pyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(3R,4R)-3-hydroxy-1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl]pyridine-4-carboxamide
6-(2-oxo-2H-chromene-3-carbonyl)-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
2-(2-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
(2S,3R)-2-amino-3-hydroxy-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
1-ethyl-3-methyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
N-{2-[(3-propanamidophenyl)formamido]ethyl}pyridine-4-carboxamide
6-ethyl-N,2-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
2-(piperidin-1-yl)-N-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide