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2-(cyclopentylmethyl)-N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[3-(1H-pyrazol-4-yl)benzoyl]-4-(pyridin-2-yl)piperazine
2-methyl-6-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]pyrimidin-4-ol
1-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-indole-3-carboxamide
2-[9-(1H-1,3-benzodiazol-2-ylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}azepane
methyl[(3-methylthiophen-2-yl)methyl][1-(pyridin-3-yl)propyl]amine
4-methylphenyl (7S,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidine-3-carbonyl]pyridine
2-(4-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
1-[2-(1,3-benzoxazol-2-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
2-(1-ethylpiperidin-4-yl)-1-[2-(3-fluorophenyl)piperidin-1-yl]ethan-1-one
2-hydroxy-3-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}-1,4-diazepan-5-one
2-(4-methyl-1,4-diazepan-1-yl)-2-[3-(2-methylpropoxy)phenyl]acetic acid
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
7-(2-methoxyethyl)-2-(1-methyl-1H-indole-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-fluorophenyl)-2-[5-(furan-2-yl)-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-5-methylpyrimidine
2-(4-chloro-2-methylphenoxy)-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
{9-[(4-methylpiperazin-1-yl)sulfonyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
6-cyclopropyl-2-{3-[(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-{2-[(3,4-dimethoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
4-ethyl-5-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
methyl 3-{imidazo[1,2-a]pyridine-2-carbonyl}-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4,6-dimethylphenol
2-[1-(2-phenylethyl)-4-(thian-4-yl)piperazin-2-yl]ethan-1-ol
1-[(2-fluorophenyl)methyl]-N-[(6-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
4-methoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
4-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)morpholine
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(4-methoxybenzoyl)piperazine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]pyridine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(propylsulfanyl)acetamide
4-[(4-fluorophenyl)methyl]-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]piperidine
(3aS,6aS)-2-(2-methoxybenzenesulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(3S,4R)-4-amino-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl]ethan-1-ol
N,6,8-trimethyl-2-(1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)ethyl]quinoline-4-carboxamide
3-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-N-(4-methylphenyl)-3-oxopropanamide
[5-chloro-7-(2-methyl-1H-imidazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-methyl-7-{2-[4-(propan-2-yl)phenyl]acetyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(benzyloxy)-1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
2-{[2-(pyrrolidine-1-carbonyl)phenyl]amino}acetic acid
6-(2,5-dimethylphenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 3-[(3S,4R)-1-[(4-hydroxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
(4aR,8aS)-1-(2-cyclohexylethyl)-6-(1,2,5-thiadiazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-[(4-chlorophenyl)methyl]-8-(3,6-dimethylpyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one