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1-{2-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-4-ol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
8-(1,3-thiazol-4-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(cyclopent-1-ene-1-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
4-(4-phenoxybutyl)-1,4-oxazepan-6-ol
N-(3,4-dimethylphenyl)-1-(3-methoxybenzoyl)piperidin-3-amine
(4aS,7aR)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,3S,6R)-5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
methyl 3-(2-cyclopropylquinoline-4-carbonyl)-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(2-fluorophenyl)formamido]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanamide
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-[(2-butyl-1H-imidazol-4-yl)methyl]-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
[(3R,4R)-1-(5-chloro-1H-indole-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,3-oxazole-5-carboxamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
(3S,5R,9R)-11-(3-chlorobenzoyl)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
3-(2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-4-(propan-2-yl)piperazin-2-one
8-cyclopropanecarbonyl-2-[(3-fluoro-2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(4-methanesulfonylphenyl)-3-(piperidine-1-carbonyl)pyridine
4-[3-(phenoxymethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]azepane
5-(2-methoxyphenoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-(ethylamino)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpyrimidine-5-carboxamide
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[4-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]methanol
(2S)-2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol
2-({[(3R,4R)-1-[(3,4-dimethylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(azepan-1-yl)-2-phenylethyl]-3-(pyridin-4-yl)propanamide
1-ethyl-4-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperazin-2-one
2-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]sulfonyl}benzoic acid
1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-cyclopropyl-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-(pyridin-2-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-ol
4-(2,2-dimethylpropyl)-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2-ethoxyethyl)-4-phenyl-1H-imidazole
1-[2-({[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}amino)ethyl]imidazolidin-2-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,2-dione
5-[(2-cyanophenyl)methyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(2-fluorophenyl)methyl]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
ethyl 5-(2,6-dimethylpyrimidine-4-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(4-fluorophenyl)ethan-1-one
N-methyl-N-(piperidin-3-ylmethyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(1H-1,2,3-triazole-5-carbonyl)pyrrolidin-3-yl]methanol
2-(carbamoylamino)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
(3aS,7aR)-5-methyl-2-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(pyridin-3-ylmethyl)-4-[4-(pyrrolidin-1-yl)benzoyl]-1,4-diazepane