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3-hydroxy-3-{[(1-methoxy-2-methylpropan-2-yl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
5,7-dimethyl-6-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-[1,2,4]triazolo[1,5-a]pyrimidine
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
ethyl 7-[4-(trifluoromethyl)benzamido]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
N-benzyl-5-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-hydroxy-2-methylbenzamide
4-(4-ethyl-5-methylpyrimidin-2-yl)-N-(4-fluorophenyl)piperazine-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylpropyl)piperidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
3-(6-methoxypyridin-3-yl)pyridin-4-amine
1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yl)ethan-1-one
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methyl-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
3-(2-chlorophenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-phenylpropanamide
(2S,4S,5R)-5-(2-chlorophenyl)-4-[(1H-imidazol-2-ylmethyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
2-methyl-6-{1-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
8-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(3-fluorophenyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
(2R,3R,6R)-5-(3-methoxybenzoyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
8-(4-chloro-2-hydroxybenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S)-2-hydroxy-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-phenylacetamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(pyridin-2-ylmethyl)pyridin-2-amine
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-[(4-benzoylpiperazin-1-yl)methyl]phenol
3-[1-(3-methoxypropanoyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
methyl 5-methyl-2-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1H-imidazole-4-carboxylate
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
2-methyl-N-(2,2,2-trifluoroethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
3-(3-fluorophenyl)-5-[5-(methoxymethyl)thiophene-2-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-amino-N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)cyclopentane-1-carboxamide
4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
(1S,4R)-2-{2-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2-azabicyclo[2.2.1]heptane
4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylate
2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylate
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(3-methoxypropyl)-N-methylpiperidine-3-carboxamide
3-[3-({[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
N-(2H-1,3-benzodioxol-5-yl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
5-{[(2,6-difluoro-3-methylphenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({4-methyl-6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-2-yl}amino)phenol
2-(3,4-dimethoxyphenyl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
[(4-methanesulfonylphenyl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[4-methoxy-3-(methoxymethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{2-[4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamido]ethyl}-1,3-thiazole-4-carboxylic acid