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(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2,2-diphenylethyl)-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
8-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
N-(2H-1,3-benzodioxol-5-yl)-5-{4-hydroxy-1-[(2-methylphenyl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
1-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]azepane
N-methyl-5-({[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1,2,4-oxadiazole-3-carboxamide
N7-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-[1,2,4]triazolo[4,3-c]pyrimidine-5,7-diamine
5-(2-methoxyphenoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(1-methyl-1H-imidazole-2-carbonyl)pyrrolidine-2-carboxamide
6-(2-chlorophenyl)-N-(2,3-dihydroxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
4-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
ethyl 5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
3-[(3-carbamoylphenyl)methyl]-N-ethylpyrrolidine-1-carboxamide
5-(2-methylphenyl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1,2,4-triazin-3-amine
2-methyl-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
1-(2-aminoethyl)-N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl}pyrimidine
4-(cyclohexylmethyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-chlorophenyl)-2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)propan-1-ol
1-{2-hydroxy-3-[3-({[3-(propan-2-yloxy)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-[(5-chloro-2-propoxyphenyl)methyl]-4H-1,2,4-triazole
6-methyl-2-[1-(7-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(5S)-5-{[benzyl({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
{[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
(2S,4R)-N-ethyl-4-(4-{[(piperidine-1-sulfonyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
4-(1H-imidazol-1-yl)-1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidine-4-carboxylic acid
N-[(2-aminopyrimidin-5-yl)methyl]-2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methylacetamide
N-[3-fluoro-5-(trifluoromethyl)phenyl]-4-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
(4aR,8aS)-1-[2-(2-methoxyphenyl)ethyl]-6-[2-(thiophen-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-5-chloro-1,2-dihydropyridin-2-one
8-[(3-chlorophenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-({1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}methyl)benzoic acid
3-(4-hydroxyphenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
1-[4-(piperidin-1-yl)benzoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzonitrile
3-cyano-5-fluoro-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
3-methoxy-1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propan-1-one
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(1H-imidazol-1-ylmethyl)piperidine
methyl 3-(2-methoxypyridine-3-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-methoxybenzoyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
N1-(5-methylpyridin-2-yl)-N3-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}propane-1,3-diamine
3-cyclopentyl-1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-{3-[methyl(phenyl)amino]propyl}urea
N-ethyl-2-(3-{3-[6-(trifluoromethyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)acetamide