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(3S,5S,9R)-5-(benzylamino)-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
6-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[2-(naphthalen-1-yl)ethanesulfonyl]pyrrolidine-2-carboxamide
1-(4-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
(3S,5S)-5-(4-methylpiperazine-1-carbonyl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(3-phenylpropyl)piperidin-3-yl]propanoate
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-(2,3-dihydro-1-benzofuran-7-yl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
N-(2-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](2-methoxyethyl)(propan-2-yl)amine
(2R,6R)-4-(1H-imidazol-2-ylmethyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-1-methyl-1H-imidazole
4-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-4-oxobutane-1-sulfonamide
1-(pyrazin-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)acetyl]-1,4-diazepane-6-carboxylic acid
6-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
(2S,4S)-4-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-methylpyrrolidine-2-carboxamide
6-[2-(2,4-dimethylphenoxy)ethyl]-N,N-dimethylpyrimidin-4-amine
(but-2-yn-1-yl)({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(furan-2-ylmethyl)amine
4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-6-(morpholin-4-yl)pyrimidin-2-amine
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
2-[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(2-phenylethyl)acetamide
4-[3-(4-fluorophenoxy)propyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-1,3-benzothiazole-5-carboxamide
2-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,2,3,4-tetrahydroisoquinoline
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
2-(5-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
3,6-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-benzofuran-2-carboxamide
N-ethyl-5-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}pyrimidin-2-amine
benzyl(methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
5-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
N-ethyl-5-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-cyclobutyl-3-{[3-(morpholin-4-yl)azetidin-1-yl]sulfonyl}benzamide
(2S,4S)-4-amino-1-[(2-tert-butylpyrimidin-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(piperidine-1-carbonyl)pyridine
2-amino-4-[2-(dimethylamino)pyrimidin-5-yl]-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-4-oxopentanamide
2-[1-benzyl-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl]ethan-1-ol
3-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
ethyl 1-ethyl-5-[2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(1H-pyrazol-1-yl)-N-[(4-sulfamoylphenyl)methyl]propanamide
N-[(1R,3R)-3-aminocyclopentyl]-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-cyclopropyl-9-[(2-propoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
N-(1-cycloheptylpiperidin-3-yl)-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine