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4-[15-methyl-9-(5-methylthiophen-2-yl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carbonyl]piperazine-1-carbaldehyde
4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]morpholine-2-carboxamide
3-(5-acetyl-2-ethoxyphenyl)-1-methyl-1-[(3-methylpyridin-4-yl)methyl]urea
5-{2-[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
(1-{[1-(2-methylquinolin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
2-(4-methoxyphenoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-4-(propan-2-yl)pyrimidine
5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
8-methoxy-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(3-methoxyphenyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
2-{5-[1-(2,6-dimethylquinoline-4-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
[(2-chloro-4,5-dimethoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
3-{2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(4aR,8aS)-6-cyclopentyl-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-(2-hydroxy-2-phenylethyl)-N-methyl-3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-[2-(trifluoromethyl)pyrimidin-4-yl]thiomorpholine
2-(4-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}phenyl)-2-methylpropanenitrile
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-methoxyethan-1-one
1-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-3-yl)acetamide
1-cyclopentyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1,2-oxazole-5-carboxamide
2-[5-(3-phenylpiperidine-1-carbonyl)-1H-pyrazol-3-yl]phenol
4-(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)benzoic acid
1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-phenylpiperidine-4-carbonitrile
8-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-methyl-1-(2-methylpropyl)-4-(3-phenylbenzoyl)piperazin-2-one
8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-[(4aR,8aR)-4a-hydroxy-7-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carboxamide
(furan-2-ylmethyl)[(6-methylpyridin-2-yl)methyl](thiophen-3-ylmethyl)amine
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(4-cyanophenyl)-1H-pyrazol-1-yl]acetamide
N-{2-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-3-carboxamide
N-[2-ethyl-1-methyl-5-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazol-7-yl]-2-methoxybenzamide
8-(2-amino-6-methoxypyrimidin-4-yl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-phenyl-4-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]pyrimidine
6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(methylsulfanyl)pyrimidin-4-amine
1,5,6-trimethyl-3-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-benzoyl-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
1-methyl-4-{1-[(2-methyl-1-benzothiophen-3-yl)methyl]pyrrolidin-3-yl}piperazine
2-(5-acetylthiophen-3-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)-1,3-oxazole
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-fluoro-3-methylbenzoyl)piperidine
4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-acetamidopyrrolidine-1-carboxamide
2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile