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ethyl 1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
methyl[(4-{2-[4-(1-methylpiperidine-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](quinolin-6-ylmethyl)amine
2-methyl-1-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]azetidin-3-yl}piperidine
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methyl-6-(propan-2-yl)pyrimidine
2-{8-benzyl-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
1,3-dimethyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N,4-dimethyl-2-(methylamino)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3-thiazole-5-carboxamide
2-(cyclopentylmethyl)-1,6-dimethyl-4-oxo-N-(quinolin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-(4H-1,2,4-triazol-4-yl)-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-[2-(2-chlorophenyl)-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2,1,3-benzoxadiazole-5-carboxamide
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amine
3-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N,N-bis(prop-2-en-1-yl)piperidine-4-carboxamide
2-{4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-ol
1-[1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-(morpholine-4-sulfonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
5-(3,5-dimethyl-1-benzofuran-2-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(2-fluorophenyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
3-(4-methyl-1H-imidazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-methoxyethan-1-one
N-[3-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]methanesulfonamide
ethyl 1-(prop-2-en-1-yl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
4-benzyl-3-ethyl-1-(4-methylpyridine-3-carbonyl)-1,4-diazepan-5-one
4-(pyridin-4-ylmethyl)-11-({[2-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{5-[1-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
4-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}morpholine-2-carboxamide
N-(3-chlorophenyl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
1-(5-chloropyridin-2-yl)-4-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidine-3-carboxylic acid
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(2-chloro-6-fluorophenyl)methyl]piperazin-2-one
(3E)-1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}hex-3-en-1-one
4-[(3-methoxyphenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
1-ethyl-3-(2-methylpropyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-pyrazole-5-carboxamide
1-{4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-[(1S,5R)-6-(1H-indol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-(benzyloxy)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(3R,4S)-4-(4-methoxyphenyl)-1-(propane-1-sulfonyl)pyrrolidin-3-amine
N-[5-({[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]carbamoyl}amino)-2-methylphenyl]propanamide
{1-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]piperidin-3-yl}methanol
(1S,5R)-3-(6-chloro-2H-chromene-3-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-carboxypiperazin-1-yl)-1-methyl-1H-1,3-benzodiazole-5-carboxylic acid
2-[4-(2-ethoxyphenyl)piperazin-1-yl]-4-(pyridin-3-yl)pyrimidine