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1-[(5-propylfuran-2-yl)methyl]-4-(pyridin-4-yl)piperazine
2-(dimethylamino)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]benzamide
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[2-(pyridin-2-yl)ethyl]amine
4-(4-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
1-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}isoquinoline
8-[2-(oxolan-3-yl)ethyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-methoxyphenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]piperidin-4-ol
2-(2-phenylethyl)-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
(isoquinolin-5-ylmethyl)(methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
4-(4-{[(5-fluoro-2-methylphenyl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
3-(2-{7-[2-hydroxy-4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
(2S,4R)-4-amino-N-ethyl-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}pyrrolidine-2-carboxamide
5-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
3-({7-[(2R)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
N-ethyl-5-[1-(2-methoxy-5-methylbenzoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-(3-{2-oxo-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethoxy}phenyl)propanamide
N-[(4-acetamidophenyl)methyl]-2-{[2-(pyridin-2-yl)ethyl]amino}acetamide
6-fluoro-N-(oxan-4-yl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-(2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-6-methyl-2,3-dihydropyridazin-3-one
6-fluoro-2-oxo-N-[2-(piperidin-1-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
(4aS,8aR)-6-(2-ethylpyrimidine-5-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
[(3-chlorophenyl)methyl]({[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl})amine
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
(3S,4S)-1-(benzenesulfonyl)-4-[benzyl(cyclobutylmethyl)amino]pyrrolidin-3-ol
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
{3-[3-(2-methoxyphenoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]propyl}dimethylamine
5-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
(3S,4S)-1-(cyclopropanesulfonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(4-{4-[2-(pyridin-2-yl)piperidin-1-yl]piperidin-1-yl}benzoyl)-1,2,3,4-tetrahydroisoquinoline
(2E)-1-(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-phenylprop-2-en-1-one
[(3R,4R)-1-(pyridin-2-ylmethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{1H-pyrazolo[3,4-b]pyridin-1-yl}-5-(pyrrolidine-1-sulfonyl)benzoic acid
2,3,6-trimethyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}quinoline-4-carboxamide
N-[(3S,4R)-1-(4-cyanopyridin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-(furan-2-carbonyl)-3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidine
4-(4-methylphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-4-carboxylic acid
N-[(2-chlorophenyl)methyl]-3-[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]propanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(1,3-thiazol-2-yl)ethyl]acetamide
2-(2-hydroxyethyl)-8-[3-(hydroxymethyl)quinolin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
[(2,4-difluorophenyl)methyl][(3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]morpholine-4-carboxamide
methyl 2-hydroxy-5-{1-[3-(hydroxymethyl)phenyl]-1H-imidazol-2-yl}benzoate
(1R,2R,6S,7S)-4-[5-(propan-2-yl)thiophene-3-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
4-benzyl-1-methyl-3-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one