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1-{[3-cyclopentyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
2-(4-ethylpiperazin-1-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2,5-dimethyl-1,3-oxazole
3-chloro-5-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydropyridin-2-one
1-(2-fluorobenzoyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-(2-ethoxynaphthalen-1-yl)acetic acid
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]urea
1-(cyclopropylmethyl)-5-[3-(1H-indol-3-yl)propanoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{1-[(3,5-dimethoxyphenyl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
1-(dimethyl-1,2-oxazol-4-yl)-3-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)urea
N-[(2-chlorophenyl)methyl]-3-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]propanamide
9-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-[(3,5-difluorophenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-(2-ethylpyrimidine-5-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-fluorophenyl)-1,4-diazepane
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-(prop-2-en-1-ylsulfanyl)propanamide
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[1-(pyridin-2-yl)propyl]amine
4-(1H-imidazol-4-ylmethyl)-1-(2-phenylphenyl)piperazin-2-one
2-{3-[2-(methylsulfanyl)ethyl]-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-[2-hydroxy-2-(2-methylphenyl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
methyl 6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrimidine-4-carboxylate
(4aS,8aR)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-{6-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridin-3-yl}ethan-1-one
(8R,9aS)-2-(3,3-diphenylpropyl)-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{2-[cyclopentyl(methyl)amino]acetyl}pyrrolidine-3-carboxylic acid
3-benzyl-8-[(3-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentanecarbonyl-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-yl)-N-(thiophen-3-ylmethyl)benzamide
3-[1-(3-phenylbutyl)piperidin-4-yl]-1,3-oxazolidin-2-one
N-benzyl-4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
1-{4-[2-(azocane-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
4-{1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}thiomorpholine
N-{1-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxy-1-oxopropan-2-yl}acetamide
8-(3-ethoxypropanoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 6-(2,5-difluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2E)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-imidazol-4-yl)prop-2-enamide
N-methyl-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
4-{2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetyl}-1-(2-phenylethyl)piperazin-2-one
6-methyl-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
3-methyl-6-[5-(5-propyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N-methyl-2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}pyrimidin-4-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-ethyl-1,2-oxazole-5-carboxamide
(3S,7S,8aS)-7-({[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-amino-6-{2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
1-(furan-3-carbonyl)-4-[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]-1,4-diazepane
2-methyl-6-(1-{[1-(pyridin-3-ylmethyl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
1-(3-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
4-[5-(cyclopentylmethyl)-3-methyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine