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N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,3-dihydro-1H-indene-1-carboxamide
2-(propan-2-yl)-1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-imidazole
5-{2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1-cycloheptylpiperidin-3-yl)-2-(2,2-dimethyl-3-oxopiperazin-1-yl)acetamide
5-cyclopropyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-1,3,4-oxadiazol-2-amine
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]quinoxaline-6-carboxamide
[(3-chlorophenyl)methyl]({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
4,5-dimethyl 1-[(3S,5S)-1-cyclohexyl-5-[(furan-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-[3-(pyridin-4-yl)propyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-(3,3-diphenylpropyl)-2-(pyrrolidin-3-yl)acetamide
N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
(3aR,6aR)-N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(1-hydroxy-2-methylpropan-2-yl)-1-{2-[2-(pyridin-2-yl)ethoxy]phenyl}urea
(3aS,7aR)-2-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-oxazolidin-2-one
(4aR,7aS)-1-propyl-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl (4aS,8aR)-6-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylate
8-(2-phenoxyacetyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[(3-methylphenyl)methyl]-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]benzamide
5,7-dimethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
4-cyclopentyl-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]pyrimidin-2-amine
4-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
4-[2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-thiazol-2-amine
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
N-(4-{[4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)acetamide
1-[6-(1,4-diazepan-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]pyrrolidin-2-one
4-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-(2-oxoimidazolidin-1-yl)benzamide
1-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}piperidine-3-carboxamide
2-{4-cycloheptyl-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-ethyl-6-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}pyrimidin-4-amine
2,3-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
4,6-dimethyl-2-oxo-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
[(2-fluoro-4-methoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
6-(thiophen-2-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N,5-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indazole-3-carboxamide
2-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-1,3-benzodiazole
1-(cyclopropylmethyl)-3-hydroxy-3-({[(4-phenyloxan-4-yl)methyl]amino}methyl)piperidin-2-one
N-cyclopentyl-4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-4-oxobutanamide
4-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-5-methylpyrimidin-2-amine
3-{[(5-fluoro-2-hydroxyphenyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2,8-dimethylquinoline
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(piperidine-1-sulfonyl)benzamide
1-(3-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
4-{2-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}phenol
2-(2-methoxyethyl)-8-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-propoxyethan-1-one