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N-methyl-3-(propan-2-yl)-N-(quinoxalin-2-ylmethyl)-1,2-oxazole-5-carboxamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)amine
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-[(3-chloro-4-ethoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
4-(1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)morpholine
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl][(8-methoxyquinolin-2-yl)methyl]methylamine
N-[(3R,4R)-3-hydroxy-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidin-4-yl]pyrazine-2-carboxamide
4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-methyl-1,3-benzoxazole-6-carboxamide
1-{4-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-4-oxobutyl}piperidin-2-one
N-(2-chloro-6-methylphenyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[(4-methyl-1H-imidazol-2-yl)formamido]methyl}benzoate
N-(6-methoxyquinolin-8-yl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
1-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
5-chloro-3-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
2-ethyl-9-(5-methyl-1,3-oxazole-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-ylmethyl)pyridin-2-amine
3-methyl-2-({2-[1-(propan-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(1-ethyl-1H-pyrazole-3-carbonyl)spiro[azepane-4,2'-chromene]
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-4-[3-(methylsulfanyl)phenyl]benzamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(3-hydroxyphenyl)piperazin-1-yl]ethan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
1-(cyclohexylmethyl)-5-{[2-(diethylamino)ethyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
2-({2-[(3-methoxypiperidin-1-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-6-methylpyridine
4-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2,4-dichlorophenoxy)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
methyl 2-(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
methyl (2R,4S)-4-hydroxy-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidine-2-carboxylate
6-chloro-N-[(2-ethoxypyridin-3-yl)methyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
3-(2-chlorophenyl)-1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidine
11-{[(3-fluoro-4-methylphenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
6-methyl-2-(3-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]cyclohexanecarboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)propanamide
7-[2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(3S,4R)-1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3,3-dimethyl-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-4-(morpholin-4-ylmethyl)piperidin-4-ol
(4-{[(6-methoxypyrimidin-4-yl)(methyl)amino]methyl}oxan-4-yl)methanol
1-[(3-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-(2-methylphenyl)pyrimidin-5-yl]methyl})(oxolan-2-ylmethyl)amine