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3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
1-[(2-fluorophenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-2-(4-fluorophenyl)piperidine
4-{4-[(4-fluoro-2-methylphenyl)methyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(1-methylpyrrolidin-2-yl)acetamide
(1R,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[(isoquinolin-5-yloxy)methyl]-N-(oxan-4-ylmethyl)-1,3-oxazole-4-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(2H-1,2,3-benzotriazol-2-yl)-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]acetamide
4-[4-(2-propoxyethyl)piperazin-1-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
(1s,4s)-4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}cyclohexan-1-ol
N-(2-methoxyethyl)-1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-[4-fluoro-3-(trifluoromethyl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-(1H-indol-5-yl)pyridine-2-carbonitrile
1-(1-{6-[4-(dimethylamino)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
1-cyclobutanecarbonyl-N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
4-{5-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
N-methyl-4-(4-methylphenyl)-N-(2-methylprop-2-en-1-yl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
4-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-2-phenylpyrimidine
(1R,5S,8S)-N-{3-[(dimethylsulfamoyl)amino]phenyl}-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
4-(cyclohex-3-en-1-ylmethyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-amino-3-(2,4-dimethoxy-3-methylphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[(2,4-dihydroxyphenyl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-[(2-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1-propanoylpiperidine-3-carboxamide
N,5-dimethyl-2-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazole-4-carboxamide
(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
N4-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(3-methoxyphenyl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
3-{[(5-cyclopentylthiophen-2-yl)methyl](methyl)amino}propane-1,2-diol
N-[(4-chloro-2-fluorophenyl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
1-(pyridin-3-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
(2R,3R,6R)-N-cyclopentyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-chloro-5-acetamido-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
1-{4-[4-(3-propylpyrrolidin-1-yl)piperidin-1-yl]phenyl}pyrrolidin-2-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
3-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
N-(3,5-dimethylphenyl)-3-[2-(3-methoxypropyl)piperidin-1-yl]-3-oxopropanamide
2-(naphthalen-2-yloxy)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-[4-(ethylamino)pyrimidin-2-yl]-N-methylpyrrolidine-3-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-(furan-2-carbonyl)-6-azaspiro[2.5]octane
2-(1,4-oxazepan-4-yl)pyridine-3-carboxamide
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-fluorobenzamide
N-{1-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide