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1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(4aS,7aR)-1-[(3,4-dimethylphenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
5-(hydroxymethyl)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}furan-2-carboxamide
2-(2-methoxyethyl)-9-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}phenyl)propanoic acid
3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,3,6-trifluorophenyl)methyl]piperidine
7-fluoro-3-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)-1,2-dihydroquinolin-2-one
1-(2-methoxy-5-{[(3-methoxypropyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-4H-1,2,4-triazole
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
N-ethyl-2-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-1H-1,3-benzodiazole-6-carboxamide
({4-ethyl-5-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-(2,3-dihydro-1H-inden-2-yl)-4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1,4-diazepane
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[3-(propan-2-yloxy)propyl]pyrimidin-2-amine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-methoxypyrimidine
(1R,2S,9R)-11-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-cyclopentyl-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-{1-methyl-4-[(2-methylpyrimidin-5-yl)methyl]piperazin-2-yl}ethan-1-ol
5-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-4-(piperidin-1-yl)butanamide
N-cycloheptyl-2-(4-hydroxypiperidin-1-yl)-6-(3-methylphenyl)pyridine-3-carboxamide
(3aR,7aS)-5-methyl-2-(6-methylpyridine-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-(1-benzylpyrrolidin-3-yl)-3-(1-methanesulfonylpiperidin-4-yl)propanamide
1-[1-(1-benzoxepine-4-carbonyl)azetidin-3-yl]-2-methylpiperidine
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-indole-2-carboxamide
2-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-1H-1,3-benzodiazole-5-carboxamide
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
N-methyl-N-[2-(oxan-2-yl)ethyl]-3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propanamide
(2S,4R)-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-(3-methoxyphenoxy)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidine
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
7-(cyclopropylmethyl)-2-(2-methyl-1,3-benzothiazole-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-(1-propylpiperidin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-fluoro-2-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]phenol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(quinolin-3-ylmethyl)acetamide
5-methyl-3-(3-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,2,4-oxadiazole
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
3-(4-methoxy-2-methylbenzoyl)-1-(3-methylbenzenesulfonyl)piperidine
1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
(4S)-1-(3-chloro-4-methoxybenzoyl)-3,3,4-trimethylpiperidin-4-ol
1-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(propan-2-yl)urea
N-(5-acetyl-2-methoxyphenyl)-2-(4-fluorophenyl)morpholine-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]butanamide
4-fluoro-N-(2-{[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}ethyl)benzamide
methyl 3-hydroxy-2-{5-[2-methoxy-5-(propan-2-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propanoate
5-{1-[(4-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
(2S,4R)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-[2-(pyridin-4-yl)acetamido]pyrrolidine-2-carboxamide