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N-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-yl]pyridin-2-amine
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-phenylbutanamide
3-[(1-methyl-1H-indol-3-yl)methyl]-3,9-diazaspiro[5.5]undecane
5-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
7-(cyclobutylmethyl)-2-[(3-hydroxy-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-(2-{[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]formamido}ethyl)benzoic acid
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(ethanesulfonyl)piperidine
1-methyl-3-(3-{5-methylthieno[2,3-d]pyrimidin-4-yl}phenyl)-1H-pyrazole
9-(4-methoxy-3-methylbenzoyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
4-chloro-3-{1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-indazole
1-(2-methylpyridin-4-yl)-4-[4-(propan-2-yl)benzoyl]-1,4-diazepane
3-(3-methoxyphenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]-1H-pyrazole-4-carboxamide
1-(4-methoxyphenyl)-4-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]butane-1,4-dione
1-(2-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[(4-chlorophenyl)methyl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-5-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
2-tert-butyl-1-(2,3-dihydro-1H-inden-2-yl)-1H-imidazole
5,6-dimethoxy-2-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydroisoquinolin-1-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-(3-fluorophenyl)-3-{1-[1-(2-phenylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
9-[2-(methylsulfanyl)pyridine-3-carbonyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1R,3R)-3-aminocyclopentyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(2S,4R)-N,N-diethyl-1-methyl-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetamido]pyrrolidine-2-carboxamide
2,3-dimethyl-N-{[4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
7-cyclohexyl-2-(2-methyl-6-propylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-6-(1H-indol-3-yl)pyridine-3-carbonitrile
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-methyl-4-{4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-3-ylmethyl)amine
(3S,7S)-5-(piperidine-1-sulfonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-3-carboxylic acid
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
5-(4-methoxyphenyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
6-methoxy-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-{[(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
5-acetyl-6-methyl-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
8-(6,6-dimethyl-5-oxothiomorpholine-3-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
5-cyclopropanecarbonyl-1'-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[(3-methylthiophen-2-yl)methyl]cyclopentanamine
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(1S,6R)-9-[3-(1H-indol-3-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methylquinoxaline-5-carboxamide
8-(3-methylbenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
2-(4-fluorophenoxymethyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
9-(4-methylpyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-chloro-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylimidazo[1,2-a]pyridine-3-carboxamide