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N2-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-methylpyrimidine-2,4-diamine
7-[(4-fluorophenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 2-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}acetate
(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1,2-dimethyl-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-indol-5-ol
4-(2-methoxyphenoxy)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylic acid
2-methoxy-N-{7-methoxy-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl}acetamide
4-(1H-imidazol-1-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)benzamide
(2R)-2-amino-N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-3-(1H-indol-3-yl)propanamide
(3R,4S)-1-[2-(1H-imidazol-2-yl)benzoyl]-4-phenylpyrrolidin-3-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4-sulfamoylbutanamide
3-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-1,5-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(methoxymethyl)piperidine
2-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
ethyl 1-(2,3-dihydroxypropyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
6-(4-chlorophenyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperazine-1-carboxamide
2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
ethyl 4-{2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
N-(3-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-yl)acetamide
3-chloro-N-cyclopropyl-4-fluoro-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzothiophene-2-carboxamide
2-(3-methoxypropyl)-8-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-methyl-1-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)butan-1-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-(2-{[3-(dimethylsulfamoyl)-5-{[(3-methylphenyl)methyl]amino}phenyl]formamido}ethyl)acetamide
3-(cyclopropylsulfamoyl)-5-(furan-3-yl)benzoic acid
1-methyl-4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
4-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
1-(2-{4-amino-6-[(4-methylphenyl)amino]-1,3,5-triazin-2-yl}phenyl)ethan-1-one
2-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-3-methoxyphenol
(2S,4R)-4-(2-chlorobenzamido)-N-ethyl-N-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
2-[1-(2,5-dimethylphenyl)-5-(1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
3-propyl-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)urea
N-methyl-2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
3-{2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}-4,5,6,7-tetrahydro-2H-indazole
1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-2-phenylethan-1-ol
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
4-[(2-methylphenyl)methyl]-1-(thiophen-2-ylmethyl)-1,4-diazepan-5-one
methyl[(1S)-1-[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl]amine
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-4-carboxamide
N-[2-(2-ethoxyphenoxy)ethyl]-N-methyl-2-(methylsulfanyl)pyridine-3-carboxamide
3-(2,6-dimethoxyphenyl)-5-[(1-methyl-1H-pyrrol-3-yl)methyl]-1,2,4-oxadiazole
1-ethyl-3-(propan-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
2-({2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(1R,5S,8S)-8-methoxy-N-(2-methoxy-5-phenylphenyl)-3-azabicyclo[3.2.1]octane-3-carboxamide
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(dimethyl-1,2-oxazol-4-yl)benzamide