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6-ethyl-1-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-butyl-N,5-dimethyl-1H-pyrazole-4-carboxamide
4-(1-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-yl)pyridine
1-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-4-(thiophen-2-ylmethyl)piperazine
4-cyclopentyl-N-{3-[(2-methylpropyl)carbamoyl]phenyl}piperazine-1-carboxamide
[(3R,4R)-1-(3,4-dichlorobenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
methyl (2S,4R)-1-[(2,4-dimethylphenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
2-benzyl-8-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[1-(2,5-dimethylpyrimidin-4-yl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
2-methyl-1-{[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}-1H-1,3-benzodiazole
5-methyl-4-({[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
2-({1-[(2-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}formamido)-N-methylacetamide
4-{[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}pyrimidine-5-carboxylic acid
5-butyl-4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
(3R,4R)-3-hydroxy-N-[(4-methoxyphenyl)methyl]-3,4-dimethylpyrrolidine-1-carboxamide
2-methoxy-1-[(1R,5S,6R)-6-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
2-(adamantan-1-ylsulfanyl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
(3S,4R)-1-(1H-indole-2-carbonyl)-3-methoxypiperidin-4-amine
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1,2-oxazole-4-carboxamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(3-methoxypropyl)benzamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}propanamide
N-[2-(azepan-1-yl)-2-phenylethyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(1H-indol-3-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
2-tert-butyl-6-(4-chloro-3-fluorobenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-{5-[(2-chlorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
(3S,4S)-1-[(5-chlorothiophen-2-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
(1R,3S)-3-ethoxy-7-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-7-azaspiro[3.5]nonan-1-ol
1-cyclopentanecarbonyl-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-4-carboxamide
1-[1'-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-methyl-1-[1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)azetidin-3-yl]piperidine
1-(5-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
3-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)-1,2-oxazole-5-carboxamide
4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(2,5-dimethylfuran-3-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
7-[(3,4-difluorophenyl)methyl]-2-(thiophen-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-methoxy-N-[2-(2-phenoxyethoxy)phenyl]pyrrolidine-1-carboxamide
3-phenyl-1-[1-(pyridazine-3-carbonyl)piperidin-4-yl]propan-1-ol
6-methyl-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2-propylpyrimidin-4-amine
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidine
3-cyclopropyl-6-(phenoxymethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-(2-hydroxyethyl)-4-(5-methylfuran-2-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
1-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-pentylurea
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
5-ethyl-N-methyl-N-(quinolin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine