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N-(2,3-dihydro-1H-inden-5-yl)-2-(2-methoxyphenyl)pyrrolidine-1-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2,2-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)cyclopropane-1-carboxamide
3-chloro-5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]aniline
2-{4-[2-(hydroxymethyl)phenyl]phenyl}-N,N-dimethylacetamide
1-(4-{ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
2-[(1S,5R)-3-(1H-indazole-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(5-fluoro-2-methoxybenzoyl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine
2-{4-[(2S)-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
4-(pyridin-2-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidin-2-amine
1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
5-(5-chloro-2,4-dimethoxyphenyl)-1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
4-[4-(6-cyclopropylpyrimidin-4-yl)piperazine-1-carbonyl]morpholine
{[4-ethyl-5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
(1R,5R)-N-benzyl-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl (2S,3S)-2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-methylpentanoate
2-methyl-4-[4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenyl]butan-2-ol
4-(1H-imidazol-1-ylmethyl)-1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]piperidin-4-ol
2,6-difluoro-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-3-methoxybenzamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-cyclopropylpropan-1-one
2-{3-[4-(1H-1,2,3-benzotriazol-1-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2,3-dimethoxy-N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}benzamide
N-{4-[2-amino-3-cyano-5-methyl-6-(propan-2-yl)pyridin-4-yl]phenyl}acetamide
2-(5-{2-[(dimethylamino)methyl]phenyl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl)ethan-1-ol
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(4-fluorophenyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine
7-(cyclohexylmethyl)-2-[3-(1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-(3,4-dimethylphenyl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2H-1,3-benzodioxole-5-carboxamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
2-(3-cyano-2-methoxypyridin-4-yl)benzoic acid
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
3-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]phenol
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-5-methylthiophene-2-carboxamide
2-(carbamoylamino)-N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)acetamide
N-butyl-1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
(1R,5R)-3-(2,8-dimethylquinoline-4-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[2-(4-methoxybenzenesulfonamido)ethyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
8-(1-benzofuran-2-ylmethyl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(3,5-dimethyl-1H-pyrazol-4-yl)-N2,N2-diethylpyrimidine-2,4-diamine
N-benzyl-5-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)pyrimidin-2-amine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]acetamide
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-methoxy-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)pyridine-3-carboxamide