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1-cyclohexyl-N3-[(3,5-difluorophenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
3-cyclopentyl-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-[1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butane-1,2-dione
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-cyclohexanecarbonyl-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
8-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoline
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(1H-indol-4-ylmethyl)acetamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-propoxyethan-1-one
1-{6-[4-(morpholine-4-carbonyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-methyl-1H-indol-1-yl)propanamide
4-(cyclohexylmethyl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-ethyl-2-methyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]quinoline-4-carboxamide
2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-(6-methoxyquinolin-8-yl)-2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
3-[N-methyl-1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]propanamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-6-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(2-methoxyethyl)-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(5-ethyl-1,3-oxazole-4-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2E)-3-(2-chlorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]prop-2-enamide
7,8-dimethyl-2-(2-methylpyrimidin-5-yl)-4-(piperidine-1-carbonyl)quinoline
4-[1-(2,2-diphenylethyl)azetidin-3-yl]morpholine
N-(2H-1,3-benzodioxol-5-yl)-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
3-(4-phenyl-1H-pyrazol-5-yl)-1-(propan-2-yl)piperidine
2-({[4-(methylsulfanyl)phenyl]methyl}(oxolan-3-ylmethyl)amino)ethan-1-ol
6-{4-[(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyridine-3-carbonitrile
(3aR,6aR)-2-[(2-chloro-5-fluorophenyl)methyl]-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-chlorophenoxy)-1-(2-acetamidoacetyl)piperidine-4-carboxylic acid
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
1-(4-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
2-(2,5-dimethoxyphenyl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methylpyridine-3-carbonitrile
2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-1,3-thiazole-4-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-methanesulfonylacetamide
(3S,4S)-4-{methyl[(3-methylpyridin-2-yl)methyl]amino}-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
6-[(dimethylamino)methyl]-N-(4-methyl-2-oxo-2H-chromen-7-yl)-1,4-oxazepane-4-carboxamide
(oxolan-2-ylmethyl)(thiophen-3-ylmethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
2-[(3,4-dimethoxypyridin-2-yl)methyl]-2-azaspiro[4.5]decan-3-one