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1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[(3,5-dimethylphenyl)methyl]-4-(1H-indol-5-ylmethyl)piperazin-2-one
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-(pyridin-4-yl)piperazine
4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}pyrimidine
2-{[(1-benzyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}-5-methyl-1,3,4-thiadiazole
(1S,6R)-9-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(2,6-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
methyl 6-{4-methyl-3,7-dioxo-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinolin-9-yl}pyridine-2-carboxylate
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[2-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
4-({5-[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,1-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(3-methylbutyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-3-yl}propanamide
(3R,5S)-5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-3-ol
5-{[(2-methoxyphenyl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(1-{6-[2-(hydroxymethyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1,4-oxazepan-6-ol
N,N,5-trimethyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyrimidin-4-amine
1-[4-(2,2-dimethylmorpholine-4-carbonyl)phenyl]imidazolidine-2,4-dione
1-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-methyl-2-oxo-8-{[2-(propylamino)pyrimidin-5-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-butoxy-N-[3-(2-phenylacetamido)phenyl]acetamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}amine
4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}benzonitrile
1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
methyl 4-({[(3S,5S)-5-{[2-(2H-1,3-benzodioxol-5-yl)ethyl]carbamoyl}-1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl]amino}methyl)benzoate
1-[2-(phenylsulfanyl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}cyclopropan-1-amine
5-(methoxymethyl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
1-{4-[(5-ethylpyridin-2-yl)methyl]piperazine-2-carbonyl}-4-methylpiperazine
6-{1-[(1-methyl-5-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
{2-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}urea
2,2-dimethyl-5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}thiomorpholin-3-one
2-({4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-1,3-benzothiazole
N-(cyclohex-1-en-1-ylmethyl)-3-(2-methyl-1H-imidazol-1-yl)butanamide
2-(5-fluoro-2-methylphenyl)-1-(4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)ethan-1-one
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
3-(1,4-dioxan-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-methyl-N-[2-(morpholin-4-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(propan-2-yl)acetamide
N-[3-(3-fluorophenyl)phenyl]-1-(isoquinolin-5-ylmethyl)piperidine-4-carboxamide
3-(1-propyl-1H-1,2,4-triazol-3-yl)-1-(2,2,6,6-tetramethylpiperidin-4-yl)urea
4-(benzyloxy)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]butan-1-one
(2S,4R)-N,N-diethyl-1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-4-propanamidopyrrolidine-2-carboxamide
1-(1H-indole-5-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol