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6-[(4-methanesulfonylphenyl)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(2S,4S)-4-amino-1-(2,2-dimethylpent-4-en-1-yl)-N,N-diethylpyrrolidine-2-carboxamide
N-(3-methoxypropyl)-6-[4-(pyridin-4-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-methyl-6-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-2-carboxamide
{4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1,4-oxazepan-6-yl}methanol
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(pyrrolidin-1-yl)propan-1-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
{[(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-[(diethylcarbamoyl)methyl]-1H-1,2,3-triazole-4-carboxamide
8-[(4-methylnaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-methyl-N-[(4-phenylphenyl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(naphthalen-2-yloxy)propanamide
1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-3-(1H-pyrazol-5-yl)piperidine
3-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-(1-methyl-1H-pyrazol-5-yl)-2-{3-[2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
5-cyclopropanecarbonyl-1'-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-3-acetamidobutanamide
1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
2-(2-benzyl-1,3-benzoxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-[(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)methyl]furan-2-carboxamide
2-methoxy-N-({3-methyl-7-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-phenylacetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}propanamide
N-(5-oxo-1-propylpyrrolidin-3-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(cyclohexylmethyl)-4-(1H-imidazol-4-ylmethyl)morpholine
6-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxylic acid
1-{1-ethyl-5-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
9-[(2S)-2-amino-2-phenylacetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)thiophen-2-yl]ethan-1-one
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]urea
2-methyl-4-{3-[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl[(1-methyl-1H-imidazol-2-yl)methyl]({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
(1R,5S,6R)-3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
1-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-3-[1-(2,5-difluorophenyl)cyclopropyl]urea
1-(1-benzylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-3-carboxamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-6-methoxyphenol
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{3-[2-amino-3-cyano-6-(2,5-dimethylfuran-3-yl)pyridin-4-yl]phenoxy}acetamide
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyridin-3-yloxy)piperidin-1-yl]propan-1-one
{[4-ethyl-5-(1-methylpiperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(furan-2-ylmethyl)[1-(4-methoxyphenyl)ethyl]methylamine
1-(2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidine-3-carboxamide
ethyl 2-{1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]piperidin-2-yl}acetate
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-methyl-6-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,6-dihydropyridine-3-carboxamide
9-methyl-3-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-3,9-diazaspiro[5.6]dodecan-10-one