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(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(pyridin-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(1S,5R)-3-[3-(2,3-dihydro-1H-isoindol-2-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-chlorophenyl)-1-(cyclopropylmethyl)-6-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]amine
3-[(1-ethylpyrrolidin-2-yl)methyl]-1-(6-phenoxypyridin-3-yl)urea
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-butyl-7,8-dimethyl-N-(propan-2-yl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(thiophen-3-yl)acetyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
[(3R,4R)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-({3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-3-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(5-methyl-1,3-oxazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
5-methanesulfonyl-1'-[(2S)-pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-{1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
(3S,4R)-1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-6-azaspiro[2.5]octane-1-carboxamide
2-(2-methyl-1H-indol-3-yl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
5-{[1-(2-chlorophenyl)cyclopropyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-benzyl-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[(4-hydroxyphenyl)methyl]-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)propanamide
3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-(propan-2-yl)propanamide
1'-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]oxolane-3-carboxamide
(2S,4S)-N-ethyl-1-[(3-hydroxyphenyl)methyl]-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
N-cyclopropyl-2-(1H-1,2,3,4-tetrazol-5-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
1-cyclohexyl-4-[3-(1,2-oxazinan-2-yl)propanoyl]piperazin-2-one
5-cyclopropyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,2-oxazole-3-carboxamide
(3S,4S)-1-{1-[(3,4-dimethylphenyl)amino]cyclohexanecarbonyl}piperidine-3,4-diol
6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-(1-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-methyl-9-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
2-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
6-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-2-methyl-1,4-diazepan-5-one
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
ethyl 3-benzyl-1-(dimethylsulfamoyl)piperidine-3-carboxylate
3-(4-hydroxyphenyl)-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-phenylpropan-1-one
methyl[(4-{[1-(naphthalene-2-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl](quinolin-6-ylmethyl)amine
5-methyl-1-(4-{4-[(1-methylpiperidin-4-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
1-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}imidazolidin-2-one
2-{[(6-methoxypyrimidin-4-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(4aS,7aR)-1-(2-fluorobenzoyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione