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7-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-methyl-N-(1-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-2-phenylethyl)thiophene-3-carboxamide
{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}(methyl)(pyridin-4-ylmethyl)amine
N-(2-methoxyethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
N-cyclopentyl-2-(dimethyl-1,2-oxazol-4-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)acetamide
4-[4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]but-3-yn-1-ol
2-methyl-7-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-[1-(propan-2-yl)piperidine-4-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
[(3R,4R)-1-[4-(difluoromethoxy)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-methoxypyrimidine-5-carboxamide
2-{4-[(4,5-dimethylfuran-2-yl)methyl]morpholin-3-yl}acetic acid
2-{4-[(2-fluorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
[2-({4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperazin-1-yl}methyl)phenyl]methanol
N-[(2,4-dimethoxyphenyl)methyl]-4,6-dimethylpyrimidin-2-amine
4-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-2-(trifluoromethyl)morpholine
4-benzyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-one
4-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
(2S)-4-methanesulfonyl-2-{[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]formamido}butanoic acid
(4aS,7aR)-1-[(3-fluoro-5-methylphenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(carbamoylmethyl)-N-[2-(2,4,6-trimethylphenoxy)ethyl]piperidine-3-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-[(1S,2R)-2-aminocyclobutyl]-2H-1,3-benzodioxole-5-carboxamide
1-methyl-N-[(2-methyl-1,3-oxazol-4-yl)methyl]-N-(2-phenylethyl)piperidin-4-amine
2-({2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
1-{5-[3-butyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
(3S,4S)-4-(propan-2-yloxy)-1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-ol
1-(2-phenylethyl)-3-(propan-2-yl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5,6-dimethyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-(2-methylpropyl)piperidine
2-(3,4-dichlorophenyl)-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
N-{[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
2-({4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
2-[4-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)piperidin-1-yl]pyridine-3-carbonitrile
N-(5-propyl-1,3,4-oxadiazol-2-yl)-1-(pyrrolidine-1-carbonyl)piperidin-4-amine
ethyl 4-(5-phenyl-1,2-oxazole-4-amido)piperidine-1-carboxylate
(4aR,7aS)-1-cyclopropanecarbonyl-4-[3-(3-fluorophenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]methyl}phenol
7-fluoro-1-(pyridin-2-ylmethyl)-3-({[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-(1-methyl-1H-pyrazol-5-yl)-2-[5-(quinolin-8-yl)-1H-indazol-1-yl]acetamide
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(piperidin-1-yl)piperidine
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
1-(3-hydroxy-2,2-dimethylpropyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-[5-(4-methyl-1H-imidazol-5-yl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl]butan-2-ol