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(2R,3S,6R)-3-(4-methylphenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-oxoethyl}acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
5-[({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]-N-methylfuran-2-carboxamide
4-chloro-5-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-methyl-1H-pyrazole
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
4-chloro-N-(furan-2-ylmethyl)-1,5-dimethyl-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
5-(2,3-difluoro-6-methoxyphenyl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
3-(1-cycloheptylpiperidin-3-yl)-1-(3,4-dimethoxyphenyl)urea
7-(2-methoxyethyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-(methoxymethyl)-N-(1,2-oxazol-3-ylmethyl)thiophene-2-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
1-(4-{[3-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)oxane-2-carboxamide
1-tert-butyl-4-[4-(2-methylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-4-methylbenzamide
1,3-dimethyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{[(1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-[(2-chlorophenyl)methyl]-4-[4-(2,2-dimethylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)pyrazine-2-carboxamide
(1S,5R)-6-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyrrolidin-1-yl)ethyl}pyridine
(1H-1,3-benzodiazol-2-ylmethyl)({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
9-acetyl-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-1'-[(5-phenylthiophen-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(3-fluorophenyl)-4-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}piperazin-2-one
4-[5-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(2-methoxyethoxy)ethan-1-one
N-methyl-1-(1-methylpiperidin-4-yl)-N-[(5-propyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
5-[2-(1H-pyrazol-1-yl)butanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
methyl 3-[(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}phenyl)formamido]propanoate
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
2-[({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]pyridine-3-carboxamide
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
4-(2,3-dihydro-1H-isoindol-2-yl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]butanamide
7-(5-chloropyridin-2-yl)-4-(1-methyl-1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
(2S,4R)-N-ethyl-1-[(3E)-hex-3-enoyl]-4-(3-hydroxybenzamido)pyrrolidine-2-carboxamide
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-[({1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}oxy)methyl]pyridine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-(4-fluorophenyl)pyrrolidin-1-yl]propan-1-one
(2S,4S)-4-amino-N-ethyl-1-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]pyrrolidine-2-carboxamide
2-(4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
[(2S)-1-[3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzoyl]pyrrolidin-2-yl]methanol
(3aS,6aS)-2-(cyclopropylmethyl)-5-(1,4-dithiepan-6-yl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(3-methoxybenzoyl)-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-cyclopentyl-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one