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N,1-dimethyl-N-[(2-methylpyridin-4-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3,7-trimethyl-1H-indole
2-butanoyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[3-(pyrrolidin-1-yl)propyl]amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-methoxy-N-methylquinoline-4-carboxamide
2-[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
7-{[4-(4-amino-5-methylpyrimidin-2-yl)piperazin-1-yl]methyl}-4-methyl-2H-chromen-2-one
2-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}benzoic acid
1-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(propan-2-yl)-1H-imidazole
(3S,4R)-4-(3-methoxyphenyl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)amino]-N-(1,3-thiazol-2-yl)acetamide
6-(piperazin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-2-(pyridin-3-yl)morpholine
3-(3-fluorophenyl)-6-[(3-hydroxyphenyl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-[3-(2-chlorophenyl)-5-methyl-1,2-oxazol-4-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-benzyl-1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl]-3-methoxy-2,2-dimethylpropanamide
3-(3-fluoro-4-phenylbenzoyl)piperidine
N-methyl-N-[3-(oxolan-2-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-chloro-2-(oxolan-3-ylmethyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
5-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-{5-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[4-(3-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}acetamide
1-[4-phenyl-1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethan-1-one
N-(2H-1,3-benzodioxol-4-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-amino-4-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(1-hydroxy-3-methylbutan-2-yl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(3R,4R)-4-cyclopropyl-3-methyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-ol
(3S,9aR)-3-(4-aminobutyl)-8-(quinolin-8-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
2-{[2-(pyridin-3-ylformamido)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2-{4-[(dimethylamino)methyl]thiophen-2-yl}-1H-imidazol-1-yl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,3-thiazole
2-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-phenylpyrimidine-5-carboxamide
[(6-chloropyridin-3-yl)methyl](isoquinolin-5-ylmethyl)methylamine
N-cyclopropyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
4-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]amine
1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-4-(2-ethoxyethyl)-1,4-diazepane-6-carboxylic acid