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N,N-dimethyl-4-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
1-(pyridin-3-ylmethyl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-(pyridin-4-yl)-5-[2-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]pyrimidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(2-oxoazepan-1-yl)propanamide
N3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2-(methylsulfanyl)benzamide
4,6-dimethyl-3-[4-(thiophen-3-ylmethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(7S,8aS)-7-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
methyl 1-[(3S,5S)-5-(azepane-1-carbonyl)-1-[(4-ethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-[(3-methoxyphenyl)methyl]morpholine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-(pyrazin-2-yl)piperidin-4-amine
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
1-ethyl-4-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}piperazine
2-{5-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methoxyphenol
7-hydroxy-6-methyl-4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1,2,3,4-tetrahydroquinolin-2-one
5-(2-chlorophenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]furan-2-carboxamide
1-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
1-{[3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methyl}-4-ethylpiperazine
7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
(3S,4R)-4-(2-methylphenyl)-1-(4-methylpiperidine-4-carbonyl)pyrrolidine-3-carboxylic acid
2-[2-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)ethyl]-6-phenyl-2,3-dihydropyridazin-3-one
N-(2-methyl-1-benzofuran-7-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
[(1-cyclohexylpiperidin-3-yl)methyl](2,3-dihydro-1-benzofuran-5-ylmethyl)(pyridin-3-ylmethyl)amine
1-ethyl-2-[1-(oxan-2-ylmethyl)-1H-imidazol-2-yl]-1H-1,3-benzodiazole
5-tert-butyl-2-(4-methanesulfonylphenyl)-1H-1,3-benzodiazole
6-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)-2-methylpyrimidin-4-ol
(3-{5-[(E)-2-(4-fluorophenyl)ethenyl]-4-phenyl-1H-imidazol-1-yl}propyl)(methyl)amine
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(thiophene-2-carbonyl)piperazine
2-cyclopropyl-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-5-carboxamide
1-methanesulfonyl-4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazine
7-(oxan-4-yl)-2-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethoxy}phenyl)propan-1-one
3-(2-{1-[(4-chlorophenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)pyridine
6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
(5-{1-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
dimethyl(2-{2-[1-(5-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
2-(dimethyl-1,3-thiazol-5-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]ethan-1-one
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1-{1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carbonyl}piperidin-4-yl)(phenyl)methanol
N-[(2S,4R,6S)-2-ethyl-6-[2-(pyridin-2-yl)pyrimidin-5-yl]oxan-4-yl]benzamide
2-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,8-diazaspiro[4.5]decane
7-methyl-2-[(3-methylquinoxalin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-N'-(2,4,6-trimethylphenyl)butanediamide
1-[2-(4-chlorophenyl)ethyl]-N-[2-(4-methylpiperazin-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-4-(thiophen-2-ylmethyl)piperazine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N5-[2-(methylsulfanyl)ethyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine