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4-{1-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
2-chloro-9-methyl-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
2-{2-[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrazine
1-[2-amino-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]butane-1,2-dione
3-{[(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)oxy]methyl}pyridine
2-{2-[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
4-(hydroxymethyl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}azepan-4-ol
ethyl 4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperazine-1-carboxylate
(2,2-diphenylethyl)(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-[(4-chlorophenyl)methyl]-3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
(3aR,5S,6S,7aS)-2-[(4-methoxynaphthalen-1-yl)methyl]-octahydro-1H-isoindole-5,6-diol
4-[4-(2-methyl-1H-imidazole-4-carbonyl)piperazin-1-yl]quinazoline
5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
(4aS,7aR)-1-[(4-methoxy-3-methylphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)pyridin-2-amine
1-(cyclohexylmethyl)-N,N-dimethyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[1-(1-cyclopropylethyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-3-(4-methoxyphenyl)-1H-pyrazole
1-ethyl-4-{1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}piperazine
N-[3-(oxolan-3-yl)propyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(1R,5R)-3-(pyridine-4-carbonyl)-6-(thiophen-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1,3-dimethyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(pyridin-3-ylmethyl)-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-[5-(3-methylphenoxymethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine
N-[2-(2-methoxyphenoxy)phenyl]-3-propoxypiperidine-1-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-methoxy-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(1-hydroxybutan-2-yl)-3-methyl-4-oxo-N-(pyridin-4-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
N-[2-(3-chlorophenyl)ethyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
1-[benzyl(methyl)amino]-3-{5-[(dimethylamino)methyl]-2-methoxyphenoxy}propan-2-ol
ethyl 4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
1-cyclohexyl-N3-[(2,4-difluorophenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperazine-1-carbaldehyde
2-[1-(2,2-dimethylpropyl)-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
3,6-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-benzofuran-2-carboxamide
2-amino-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(pyridin-3-yl)propanamide
1-[4-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)thiophen-2-yl]ethan-1-one
3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(2-fluorophenyl)piperidine-1-carboxamide
4-ethyl-3-{2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
1-[2-(2-butoxy-5-methylphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
3-[3-(benzyloxy)phenyl]-1-methyl-1-(oxan-2-ylmethyl)urea
2-(5-acetamido-1H-1,2,4-triazol-3-yl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)acetamide
N3-[(4-fluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-cyclopropyl-8-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-chloro-2-methoxy-6-(pyrrolidin-1-ylmethyl)phenoxy]propanoic acid