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3-[3-(oxan-4-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
2-(2-phenyl-1H-imidazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2,4-dimethoxybenzamide
3-{1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}propanamide
7-[(3,4-difluorophenyl)methyl]-2-(3,5-dimethylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[1-(morpholin-4-yl)cycloheptyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-N,N-dimethylpyrrolidin-3-amine
3-{2-[2-(3-acetyl-2,4,6-trimethylphenyl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
8-chloro-N-[(1-hydroxycyclohexyl)methyl]quinoline-2-carboxamide
N-methyl-5-[(3-methylbutyl)amino]-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(2,3-dihydro-1H-inden-2-yl)-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
3-[5-(4-ethyl-2-methyl-1,3-thiazol-5-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-methyl-1H-imidazole-2-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
N-({1-[(6-ethyl-2-oxo-2H-chromen-4-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)acetamide
N-methyl-N-(oxan-4-yl)-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
(2S)-2-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-3,3-dimethylbutan-1-ol
2-(2,3-dimethoxyphenyl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-4-(pyridin-3-yl)piperidin-4-ol
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]cyclohex-1-ene-1-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
methyl 4-{[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
2-{9-[(2-methoxy-4-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
2-(3-fluorophenyl)-N-({7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
9-[2-(morpholin-4-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N,2,8-trimethylquinoline-4-carboxamide
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroquinoxalin-2-one
11-(1H-1,3-benzodiazole-5-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
6-methyl-2-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}piperidin-3-ol
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl})amine
N-cyclopropyl-1-phenyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
3,5-dimethoxy-N-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]benzamide
4-(2,6-dimethoxypyrimidine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazine
3-{[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N-[4-(3-fluorophenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(3S,4R)-1-(2,3-difluoro-4-methoxybenzoyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-(cyclopropylmethyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2-chlorophenyl)-3-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
N-(furan-2-ylmethyl)-N,2,8-trimethylquinoline-4-carboxamide
N,1-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-benzyl-3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
4-fluoro-N-({1-[2-(4-methoxyphenoxy)acetyl]piperidin-3-yl}methyl)benzamide
1-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)ethan-1-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1-(9H-purin-6-yl)piperidin-4-amine
N-(9H-fluoren-9-yl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
methyl (2S,3S)-2-{[5-methanesulfonamido-1-(2-phenylethyl)-1H-1,3-benzodiazol-7-yl]formamido}-3-methylpentanoate