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3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-[(3,3,4-trimethylpiperazin-1-yl)methyl]piperidin-2-one
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-benzofuran-5-carboxamide
1-(1-benzofuran-3-carbonyl)-4-(1H-imidazol-4-ylmethyl)-1,4-diazepan-6-ol
2-cyclopropyl-4-hydroxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
6-fluoro-2-{[3-(morpholine-4-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
2-{3-[1-(1H-indol-5-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
1-(3-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}piperidin-1-yl)propan-1-one
(1S,2R)-N1-benzyl-N1-(2-carbamoylethyl)-N2-propylcyclohexane-1,2-dicarboxamide
N-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carboxamide
4-(3-methyl-1-benzofuran-2-yl)-1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole
2-methoxy-N-[3-({[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]carbamoyl}amino)-4-methylphenyl]acetamide
1-{2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-imidazole
4-[ethyl(4-phenylbutyl)amino]butan-1-ol
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
8-{[3-(2-aminoethyl)phenyl]methyl}-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({[(2-ethoxypyridin-3-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
N-cyclopentyl-1-(2-methylpropyl)-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-methoxy-5-methylthiophene-2-carboxamide
9-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
{[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-[(2-ethylphenyl)methyl]-4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
6-phenyl-2-{2-[(thiolan-3-yl)amino]ethyl}-2,3,4,5-tetrahydropyridazin-3-one
2-(1,3-benzothiazol-2-yl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
2,5-dioxo-6-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(3-fluorophenoxy)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
7-(5-chloropyridin-2-yl)-4-(pyrimidine-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
6-methoxy-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}pyrimidin-4-amine
4-(3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)-4H-1,2,4-triazole
[1-(cyclohex-3-en-1-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
(3aS,6aR)-3-(pyridin-2-ylmethyl)-5-[(2,3,6-trifluorophenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 1-(benzyloxy)-2-oxo-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-5-(4-methoxyphenyl)furan-2-carboxamide
4-[1-(1H-pyrazole-4-sulfonyl)piperidin-3-yl]benzoic acid
1'-[(3,4-dimethoxypyridin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aS,8aR)-1-(3-hydroxypropyl)-6-(4-methylquinolin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
2-(4-fluorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
2-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
1-ethyl-3-(morpholine-4-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
8-(1H-imidazole-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}pyrrolidine-1-carboxamide
2-[2-(dimethylamino)ethyl]-9-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one