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5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-[1'-(4-methylpyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-(2-fluorophenoxy)piperidine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(4,7-dimethylquinazolin-2-yl)azepan-4-amine
7-chloro-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
dimethyl[(4-methyl-5-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
1,3-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
3,5-dichloro-4-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)pyridine
(2E)-1-[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]-3-(1H-imidazol-4-yl)prop-2-en-1-one
N-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-[3-(2-methylpyrimidin-4-yl)phenyl]-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
N'-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)butanediamide
3-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-1-(6-methylpyridin-3-yl)urea
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(1H-indol-3-yl)ethyl]acetamide
2-(2-amino-2-methylpropanoyl)-N-(pyridin-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-5-(1-methoxypropan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(4S,6R)-N-butyl-N-(furan-2-ylmethyl)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
2-[5-cyclopropyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-fluorophenyl)pyrimidine
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}urea
5-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
(4aR,7aS)-1-{2-[methyl(2-methylpropyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-phenyl-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-5-yl}benzoic acid
7-methanesulfonyl-N,4-dimethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]quinazolin-2-amine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
(3S,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[1-(furan-2-carbonyl)piperidin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-methoxy-1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(prop-2-en-1-yl)piperidine
3-(2-fluorophenyl)-6-[3-(prop-2-en-1-yloxy)benzoyl]-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3,5-dimethoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
N-({1-[ethyl(methyl)amino]cyclopentyl}methyl)-5,6-dimethylpyrimidin-4-amine
2-{[4-(furan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(4-methoxyphenyl)-1H-imidazole
8-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-[5-cyclopropyl-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
(3aS,6aS)-2-[(2-ethylphenyl)methyl]-5-(6-methylpyridine-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({[(3R,4R)-1-(3,4-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-{1-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-{[(3S,4S)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]methyl}acetamide
3-(5-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
{3-[(3-methoxyphenyl)methyl]-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl}methanol
2-[1-methyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
5-[3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propanoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-4-(trifluoromethyl)benzamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(3,3,5,5-tetramethylcyclohexyl)piperidin-4-yl]oxy}benzamide
N-[1-(2-chlorophenyl)cyclopropyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4aR,7aS)-1-(2-methylpropanoyl)-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide