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(2S,4R)-1-benzyl-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
3-chloro-4-fluoro-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-1-benzothiophene-2-carboxamide
N-(3-methoxyphenyl)-5-(1H-pyrazol-3-yl)furan-2-carboxamide
9-(3-chloropyridin-2-yl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(adamantan-2-ylmethyl)-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
N3-(cyclohexylmethyl)-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
1-ethyl-N-(1H-imidazol-2-ylmethyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-(3-methoxybenzenesulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
13-(2-methoxypyridin-3-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
3-({ethyl[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)piperidin-3-ol
2-(3-methoxyphenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[1-(3-methoxyphenyl)ethyl]-N-methylacetamide
N-(2,2-diphenylethyl)-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-[(3S,5S)-1-(cyclopropylmethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-methanesulfonyl-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)piperazine-1-carboxamide
1-benzyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrazine
2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(4-methyl-1H-imidazol-5-yl)-4-phenyl-4H-1,2,4-triazole
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-methyloxane-2-carbonyl)piperidine
5-[2-(1H-pyrazol-1-ylmethyl)propanoyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4S)-4-amino-1-(naphthalene-1-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}acetamide
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
1-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-phenylethane-1,2-dione
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-(2-{7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
1-[1-(6-{[2-(dimethylamino)ethyl](methyl)amino}pyridine-3-carbonyl)piperidin-3-yl]-3-methylbutan-1-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
6-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-ethyl-3-methyl-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(1H-pyrazol-3-yl)piperidine
3-{1-[2-(3-methoxyphenyl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(3S,4R)-1-[(3-fluoro-5-methylphenyl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
8-(4-methyl-1H-pyrrole-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-methoxybenzoic acid
1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-5-oxopyrrolidine-3-carboxylic acid
(1R,3S)-7-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
3-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}benzonitrile
4-(3-methylphenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
N-methyl-2-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2H-chromene-3-carboxamide
N-methyl-3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-(piperidin-4-yl)benzamide
4-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]azetidin-3-yl}pyridine
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
5-chloro-N-[2-hydroxy-3-(4-methylphenoxy)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide