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(3aS,6aR)-5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N3-cyclooctyl-N5-(cyclopropylmethyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-N-[2-(propan-2-yl)phenyl]piperidine-1-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
2-(azepan-1-yl)-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
5-(1H-imidazol-2-yl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-(2-fluorophenyl)-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1,2,4-triazin-3-amine
5-(4-methanesulfonylphenyl)-4-phenyl-1-[2-(propan-2-yloxy)ethyl]-1H-imidazole
N,3,6,7-tetramethyl-N-[3-(oxolan-2-yl)propyl]-1-benzofuran-2-carboxamide
2-(propan-2-yl)-4-(1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-2-yl)pyrimidine
1-{[1-(2-carboxyethyl)-1H-pyrazol-4-yl]methyl}-3-ethylpiperidine-3-carboxylic acid
4-{[(oxolan-3-yl)carbamoyl]amino}-N-(2-phenylethyl)benzamide
3-[benzyl(pyridin-4-ylmethyl)amino]-2-methylpropan-1-ol
(2S,4S)-4-amino-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(phenylcarbamoyl)piperidin-3-yl]propanoic acid
5-[2-(benzyloxy)phenyl]pyridine-3-carboxamide
4-(3,5-difluoropyridine-2-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
N-[3-(2-methoxyphenoxy)propyl]-N-methyloxane-2-carboxamide
N-(2-methoxyethyl)-2-(1-methyl-3-oxopiperazin-2-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
2-[1-(2-chlorophenyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(furan-2-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-propyl-1H-pyrazole-4-carboxamide
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
N-[2-(dimethylamino)ethyl]-3-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)propanamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,2,3-thiadiazole-4-carboxamide
6-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-acetyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl (2S,4S)-1-[(4-chlorophenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
6-cyclopentyl-1-methyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(cyclohexylmethyl)-N-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2-[(adamantan-1-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amino]ethan-1-ol
N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
4-[4-ethyl-6-(oxolan-2-ylmethyl)pyrimidin-2-yl]morpholine
2-[4-(5,6-dimethylpyrimidin-4-yl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-[2-(1H-imidazol-1-yl)-1-phenylethyl]urea
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-(3,3,5,5-tetramethylcyclohexyl)benzamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]pyridin-2-ol
4,5-dimethyl-6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
2-amino-4-(2,6-dimethoxyphenyl)-6-(4-methyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
(1R,2R,6S,7S)-4-(dimethyl-1,3-thiazole-4-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(1H-1,2,4-triazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-2H-chromen-2-one
(1R,6S)-9-methyl-3-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]-3,9-diazabicyclo[4.2.1]nonane