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5-cyclopropyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-pyrazole-3-carboxamide
(2-methoxyethyl)[(3-phenyl-1,2-oxazol-5-yl)methyl][(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-(4-{1-[3-(trifluoromethyl)phenyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-ol
4-[3-(3-methoxyphenoxy)azetidin-1-yl]-2,6-dimethylpyridine
1-[2-(furan-2-yl)azepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-ethyl-N-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-yl}acetamide
N-[2-methyl-1-(pyridin-2-yl)propyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(3,3-dimethylbutyl)azepan-3-yl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
1-(benzenesulfonyl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
1-(oxan-4-yl)-N-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-amine
5-{[(3-chlorophenyl)methyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-methyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-N-(piperidin-4-yl)acetamide
N-[2-(2-chlorophenyl)ethyl]-2-(1-cyclopentyl-3-oxopiperazin-2-yl)acetamide
1'-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-1-[3-(methylsulfanyl)propyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N,3,5-trimethyl-N-(quinolin-8-ylmethyl)-1-benzofuran-2-carboxamide
N-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-methylpyridin-2-amine
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-3-(1H-pyrazol-4-yl)propanamide
3-(methylsulfanyl)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)propanamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-(3-methoxypropyl)-5-methyl-1H-pyrazole-4-carboxamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
N-{3-[2-(4-chlorophenyl)morpholin-4-yl]-3-oxopropyl}-N-methylmethanesulfonamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-(morpholin-4-yl)butan-1-one
2-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}quinolin-8-ol
3,5-dimethyl-4-{5-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1,2-oxazole
(3R,4S)-1-(2-fluorobenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-amine
(4-benzyl-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)methanol
4-[2-(phenylsulfanyl)acetyl]-1λ6-thiomorpholine-1,1-dione
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidine
7-(3-chlorophenyl)-4-(2-methyl-1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aR,5R,6S,7aS)-2-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
7-[2-(pyridin-4-yl)-1H-imidazol-1-yl]-2,3,4,9-tetrahydro-1H-carbazol-1-one
3-(3-hydroxyquinoxalin-2-yl)-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}propanamide
N-(2-methylprop-2-en-1-yl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-benzyl-1-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(1-ethyl-1H-1,2,3-triazol-4-yl)urea
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethoxybenzamide
2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-N-propyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
1-(4-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}phenyl)ethan-1-one
2-amino-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-methylpropan-1-one
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,1-dimethylazepane-2-carboxamide
N-[2-(6-methoxypyridin-3-yl)phenyl]cyclopropanecarboxamide
2-[3-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)phenoxy]ethan-1-ol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyrrolidine-1-sulfonyl)piperazine
[7-(2,5-dimethoxyphenyl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(2,5-dioxoimidazolidin-4-yl)acetamide
3-{[(carbamoylmethyl)(methyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide