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{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
(3S,4R)-1-{[4-(difluoromethoxy)phenyl]methyl}-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
7-chloro-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
(3R)-1-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-ol
6-methyl-2-(pyridin-3-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
3-[({2-[(2,5-dimethoxyphenyl)amino]-1,3-thiazol-5-yl}methyl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[2-(4-methoxyphenyl)ethyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-{4-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
(2R,6R)-4-(2,5-dimethylfuran-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,3-diphenylpiperidine
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]hexan-1-one
2-(2-methoxyethyl)-9-[2-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2,3-dimethylphenyl)-N,N-dimethylbenzamide
N-methyl-4-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)butanamide
5-[(2S)-2-amino-4-methylpentanoyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3-{[(4aS,7aR)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}phenoxy)acetamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-6-ethylpyrimidin-4-amine
methyl 5-[1-(oxolane-2-carbonyl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-(dimethyl-1,2-oxazol-4-yl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
1-ethyl-4-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[(3-phenyloxolan-3-yl)methyl]amine
4-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)pyridine
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
methyl 2-[({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]pyridine-3-carboxylate
N,5-dimethyl-N-(2-methylpropyl)-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2,5-dimethyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2S,4S,5R)-4-(cyclopropylcarbamoyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
(2S,4R)-N-methyl-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(2-fluorophenyl)methyl]oxane-4-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(propan-2-yloxy)acetamide
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]methyl}benzonitrile
1-cycloheptanecarbonyl-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
2-(2-hydroxyethyl)-9-[2-(4-methoxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
(2,1,3-benzoxadiazol-4-ylmethyl)({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl})(2-methoxyethyl)amine
4-methyl-5-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-amine
1-(cyclohex-3-ene-1-carbonyl)-3-(2-methoxyphenoxy)azetidine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-tert-butyl-4-hydroxypyrimidine-5-carboxamide
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
1-ethyl-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1,9-dimethyl-4-{[4-(2-methylpropyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
N-[(3S,4R)-4-(4-methylphenyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl]acetamide
(1R,5S,8S)-N-[4-(3-acetylphenyl)phenyl]-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one