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1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(thiophen-2-ylmethyl)piperazine
1-[2-methoxy-5-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
6-{[2-(dimethylamino)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-{3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propoxy}pyridine
1-cyclohexyl-3-(cyclopropylmethyl)-5-(3-oxopiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyridin-4-amine
3-(5-chloro-2-methoxyphenyl)-5-methoxypyridine
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
7-fluoro-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-2-methyl-1,4-diazepan-5-one
(3R,4S)-1-[(3,5-dimethoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
4-methoxy-N-(2-methoxyethyl)-2-({1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}oxy)benzamide
(2S,4S)-N-[2-(2-chlorophenyl)ethyl]-1-methyl-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
{4-[(1-propyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
1-[(2,5-dimethylphenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
(1R,7S)-3-tert-butyl-N-ethyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 3-cyclobutaneamido-6-({methyl[2-(4-methylphenoxy)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
(3S,4S)-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
N-{2-[1-(1-carbamoylethyl)-1,2,3,6-tetrahydropyridin-4-yl]ethyl}-2,2-dimethylpropanamide
methyl 4-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperazine-1-carboxylate
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyethoxy)ethan-1-one
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-[(3-methyloxetan-3-yl)methyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
3-[4-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-(pyridin-2-yl)piperidine-3-carboxamide
1-(1-phenylcyclohexanecarbonyl)-4-(pyrrolidin-3-yl)piperazine
2-(2-{1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-(4-{[(3S,4S)-4-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl]methyl}phenyl)acetamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
1-(pyridin-4-ylmethyl)-4-[(2,3,4-trifluorophenyl)methyl]-1,4-diazepane
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-methyl-4-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
5-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
(1R,5R)-6-(cyclopropylmethyl)-3-(5-methylpyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-5-{1-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
3-{[(4-cyanophenyl)methyl](propan-2-yl)amino}propanamide
2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
(2,3-dihydro-1-benzofuran-5-ylmethyl)({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl})(2-methoxyethyl)amine
1-[2-(azocan-1-yl)-2-oxo-1-phenylethyl]-4-butylpiperazine-2,3-dione
4-(2-fluorophenoxy)-1-(morpholine-4-carbonyl)piperidine-4-carboxylic acid
cyclopentyl 4-({[2-(ethanesulfonyl)ethyl]carbamoyl}amino)benzoate
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-3-methoxy-1,2-dihydropyridin-2-one
3-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
4-[(6-methylpyridin-2-yl)methyl]-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
3-chloro-4-({1-[(4-ethynylphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide