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2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propan-2-ol
3-[(3R,4S)-4-(dimethylamino)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-3-yl]propan-1-ol
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(4-phenoxybenzoyl)piperidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
N-[2-(dimethyl-1,3-thiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(3-hydroxyphenyl)-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
1-(5-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-ethyl-N-methyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
N-[2-(oxan-2-yl)ethyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
4-[1-(4-{5-methylthieno[2,3-d]pyrimidin-4-yl}phenyl)ethyl]morpholine
3-(3-chloro-1,2-oxazol-5-yl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
4-{2-[cyclopentyl(methyl)amino]acetyl}-1-(4-methylphenyl)piperazin-2-one
2-[4-(pyridin-4-yl)piperazin-1-yl]-4-(trifluoromethyl)pyrimidine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-[2-(3-methoxyphenyl)ethyl]piperidine
3-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethane-1,2-dione
2-[(2-fluorophenyl)methyl]-4-[4-(quinoxalin-6-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
2-(2-chlorophenoxy)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)(methyl)amino]-N-methylpropanamide
6-[(2-ethoxypyridin-3-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1S,6R)-9-[2-(pyridin-4-yl)quinoline-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-butyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
2-{4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}-4-methoxypyrimidine
(1S,5R)-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
8-{[2-(trifluoromethoxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[(1-ethyl-1H-imidazol-5-yl)methyl]-1,2-dihydrophthalazin-1-one
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(3,4-dimethoxyphenyl)methyl]piperidine
4-{4-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-1,2,3-triazol-1-yl}-N-ethylpiperidine-1-carboxamide
2-(cyclohex-1-en-1-yl)-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}acetamide
6-methyl-4-[3-(1H-pyrazol-5-yl)phenyl]-2,3-dihydropyridazin-3-one
4-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-1-(4-fluorophenyl)butan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyridine-4-carboxamide
1-(azepan-1-yl)-3-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]propan-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-(methoxymethyl)cyclopropane-1-carboxamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-3-(pyridin-3-yl)propanamide
1-[2-(6-methyl-4-oxo-3,4-dihydroquinazolin-3-yl)ethyl]piperidine-3-carboxamide
N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
4-(2-{1-[4-(methylsulfanyl)benzoyl]piperidin-2-yl}ethyl)morpholine
methyl 4-(2-methoxypyridin-3-yl)-1H-pyrrole-2-carboxylate
5-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-methyl-2-(propan-2-yl)-6-(1H-pyrazol-4-yl)pyrimidine
2-[(cycloheptylamino)methyl]-4-(pyridin-3-yl)phenol