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2-{1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}ethan-1-ol
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
3-(2-fluorophenyl)-N-methyl-3-phenyl-N-(1,3-thiazol-2-ylmethyl)propanamide
2-phenyl-7-[4-(1H-pyrazol-4-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,7-dioxo-1,3-diazepane-4-carboxamide
3-({[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}amino)-2,2-dimethylpropan-1-ol
4-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
4-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]benzonitrile
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-5-methylpyridine-3-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
1-[2-(2-methoxyphenyl)ethyl]-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
2-(2-ethoxypyridin-3-yl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
2-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-6-phenylpyridine-3-carboxylic acid
1-{3-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]phenyl}pyrrolidin-2-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-(3-chlorophenyl)-N-[4-(4-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
N-{2-[1-(3-fluorobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
3,5-dimethyl-4-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1,2-oxazole
(2S,4R)-4-amino-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-3-(trifluoromethyl)benzamide
5-benzyl-1-(4-methylphenyl)-4-(pyridazine-3-carbonyl)piperazin-2-one
[(3-{2-[4-(2,3-dihydro-1-benzofuran-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
N-(3-aminopropyl)-1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
1-[2-(3-methylphenoxy)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
2-(dimethylamino)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-6-methoxypyrimidine
N-[(3-methyloxetan-3-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-[(3S,4R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-4-propylpyrrolidin-3-yl]acetamide
4-ethyl-3-{1-[2-(quinazolin-4-yloxy)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-methoxyethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N-(2-methylphenyl)piperidine-1-carboxamide
1-benzyl-4-oxo-N3-(propan-2-yl)-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
3,5-dichloro-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,4-dimethylbenzamide
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
[1-(1H-imidazol-1-yl)propan-2-yl][(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amine
5-[4-(trifluoromethoxy)phenyl]pyrazin-2-amine
2-amino-3-ethyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-{4-hydroxy-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-N-methyl-N-(quinolin-5-ylmethyl)-1-benzofuran-2-carboxamide
4-ethyl-6-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-2-(pyrrolidin-1-yl)pyrimidine
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4-chloro-3-fluorobenzamide
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
N-[(1R,3R)-3-aminocyclopentyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(4-ethylpiperazin-1-yl)ethan-1-one