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4-[(4-methoxyphenyl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
N-({3-[(dimethylamino)methyl]-4-methoxyphenyl}methyl)-6-methoxy-1,3-benzothiazol-2-amine
N-[2-ethyl-4-(6-methyl-9H-purin-9-yl)phenyl]acetamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-fluorobenzamide
1-cyclopentyl-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
5-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-{3-[4-({[3-(trifluoromethoxy)phenyl]methyl}amino)piperidin-1-yl]phenyl}ethane-1-sulfonamide
3-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
2-(3,4-dimethoxyphenyl)-5-methyl-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}-1,3-oxazole
4-[(4-methanesulfonylphenyl)methyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
N-cyclopentyl-1-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-{5-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-(1H-pyrazole-3-carbonyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
methyl 5-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]carbamoyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylate
5-(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
2-methyl-1-(2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
ethyl 1-[(5-ethylthiophen-2-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-benzyl-2-(ethanesulfonyl)-5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
N-(2-cyclohexaneamido-5-methylphenyl)-3-methyl-1H-pyrazole-5-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-N'-cyclopentylbutanediamide
2-(1-tert-butyl-1H-pyrazol-4-yl)-6-ethyl-4-(pyrrolidine-1-carbonyl)quinoline
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
2-[1-cyclohexyl-4-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(2R,3R)-2-methoxy-1'-[3-(1,2-oxazolidin-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
8-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
6-{4-[(propan-2-yloxy)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-cyclopropyl-6-oxo-N,N-bis(pyridin-3-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
7-(3-methoxypropyl)-2-[2-(3-methylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2,5-difluorobenzoyl)-1-(thian-4-yl)piperidine
N-(3-{[cyclopropyl({[4-(methylsulfanyl)phenyl]methyl})carbamoyl]amino}-4-methylphenyl)acetamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
(2S,4R)-4-amino-N-(propan-2-yl)-1-{[1-(pyridin-4-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
methyl 3-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(4-benzylpiperidine-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
4-(4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
2-(4-chlorophenyl)-2-[methyl(1H-pyrazol-3-ylmethyl)amino]acetic acid
(3S,9aR)-3-benzyl-2-methyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-(piperidin-3-yl)pyrimidin-4-amine
{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(2-methylpropyl)amine
2-[1-(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepan-5-one
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
5-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
ethyl 4-(2-phenoxyethyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
9-methoxy-3-(2-phenoxypropanoyl)-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-[5-(3-fluoro-4-methylphenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide