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2-[4-(methylsulfanyl)phenyl]-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine
methyl 1-[(6-chloro-4-{[(2,3-dimethoxyphenyl)methyl]amino}quinazolin-2-yl)methyl]piperidine-2-carboxylate
1-[4-(1H-imidazol-1-yl)phenyl]-3-(1-methanesulfonylpiperidin-4-yl)urea
N-[(3S,4R)-1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[4-(4-methylphenyl)phenyl]piperidin-4-amine
benzyl[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl][(4-methyl-1,3-thiazol-5-yl)methyl]amine
3-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
ethyl[(4-fluoro-3-methoxyphenyl)methyl][(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-(cycloheptylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(2-phenylethyl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-(2,4-dimethoxyphenyl)-3-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)propanamide
2-methyl-4-{3-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}but-3-yn-2-ol
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N,N-dimethylacetamide
3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
[(3S,7S)-5-(5-propyl-1,2-oxazole-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
(3S,4S)-1-(2H-1,3-benzodioxol-4-ylmethyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-acetyl-8-(4-methoxy-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
6-ethoxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)ethan-1-one
3-{[(1,3-dihydroxy-2-methylpropan-2-yl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
5-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(2,3-dimethylphenyl)-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2E)-N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-3-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
N-methyl-2-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)pyridine-3-carboxamide
methyl 3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)-4-methylbenzoate
4-(1-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}ethyl)morpholine
4-{[4-(2-methylphenoxy)piperidin-1-yl]methyl}pyridine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(1-phenylcyclopentyl)methyl]acetamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
4-(benzyloxy)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
(4aS,8aR)-1-(carboxymethyl)-6-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1H-imidazol-2-ylmethyl)-4-(3-phenylpropyl)piperidine-4-carboxylic acid
(3S,4S)-1-[3-(dimethylsulfamoyl)propyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(3,4-dichlorophenyl)-4-(pyridazine-3-carbonyl)morpholine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
1-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-6-methylpyridine-2-carboxamide
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(2-phenoxyethyl)piperazine
1-(4-chlorophenyl)-N-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
methyl 3-{[5-(1H-1,3-benzodiazol-2-ylmethyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-methoxy-N-methylbenzamide
(1S,5R)-3-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-ethyl-1H-pyrazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine