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methyl 3-[(2,3-difluorophenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-methoxypiperidine
(1R,5R)-3-methanesulfonyl-6-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-3-methanesulfonyl-6-[(8-methoxy-2H-chromen-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[2-(3,4-difluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[(6-methoxynaphthalen-2-yl)methyl]pyrrolidin-3-yl]methanol
2-methyl-6-{[(2S,5R)-5-[(4-methylpiperazin-1-yl)methyl]oxolan-2-yl]methyl}quinoline
3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
N,N-dimethyl-5-{[methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]methyl}pyrimidin-2-amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyridin-3-yl)piperazin-1-yl]ethan-1-one
N-(prop-2-en-1-yl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(2-methoxyphenyl)-4-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
{[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)(pyridin-4-ylmethyl)amine
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(quinolin-5-ylmethyl)piperidin-4-ol
N,2-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2R,3R)-1'-(5-methyl-1,3-oxazole-4-carbonyl)-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-amino-4-(5-methyl-1H-indol-3-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
(1S,6R)-9-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
6-(2-phenoxyethyl)-3,4-dihydroquinazolin-4-one
2-(3-fluorophenoxymethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
(1S,5R)-N-(2H-1,3-benzodioxol-5-yl)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[4-(4-cyclohexylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(5-methylfuran-2-yl)pyrimidine
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
4-cyano-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)benzamide
(1R,2R,6S,7S)-4-(2-methyl-4-phenylpyridine-3-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3S)-3-hydroxy-3-phenylpropyl]-3-methyl-1,2-dihydroquinoxalin-2-one
6-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-2-carbonitrile
3-(3-methylthiophen-2-yl)-5-[(oxolan-2-ylmethyl)sulfamoyl]benzoic acid
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-(pyrimidin-5-yl)benzoic acid
1-(cyclobutylmethyl)-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
N-(oxolan-3-yl)-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(2-methylphenoxymethyl)piperidine
N-[(3S,4R)-1-(1,3-benzothiazol-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
9-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(pyrazin-2-yl)propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
1-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]urea
(1R,6S)-9-methyl-N-(2-methyl-5-sulfamoylphenyl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-(methylsulfanyl)pyridine
4-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]thiomorpholine
(3R,4S)-4-(5-methylfuran-2-yl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-amine
8-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3,5-dimethylphenyl)-4-[3-(1H-imidazol-2-yl)benzoyl]piperazin-2-one
5-acetyl-N-[1-(pyrazin-2-yl)piperidin-3-yl]thiophene-2-carboxamide