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N-(butan-2-yl)-2,6-difluoro-4-methoxy-N-(pyridin-4-ylmethyl)benzamide
8-(3,6-dimethylpyrazin-2-yl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(3-fluorophenoxymethyl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1,3-oxazole-4-carboxamide
4-({3-[5-(methanesulfonylmethyl)pyridin-2-yl]phenyl}methyl)morpholine
N-[(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
2-cyclopentyl-9-(thiophen-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
2-[3-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
4-[7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]benzonitrile
1-(2-ethoxyethyl)-4-(2-methyl-4-phenylpyridine-3-carbonyl)piperazine
2-(phenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
1-{4-[3-({[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
(1R,9aR)-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-octahydro-1H-quinolizine-1-carboxamide
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-cyclopentyl-2-[4-(acetamidomethyl)-5-methyl-1,2,3,6-tetrahydropyridin-1-yl]propanamide
N,5,7-trimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-methyl-1-{6-methyl-5-[5-(1-methyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}butan-1-one
7-[2-(4-phenylpyrimidin-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N,N-diethyl-1-[5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]pyrrolidin-3-amine
5-methyl-3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1,2-oxazole
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
(3S,4S)-4-methyl-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-3,4-diol
6-[(diethylamino)methyl]-N-(3-fluorophenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(2,3-difluoro-6-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-3-(2-phenylethyl)-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-(quinolin-8-ylmethyl)piperidin-4-ol
2-{N-methyl-1-[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}-2-(pyridin-3-yl)acetic acid
methyl 4-{5-methyl-4-[(3-phenylpiperidin-1-yl)methyl]-1,3-oxazol-2-yl}benzoate
2-benzyl-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
1-{4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
4-[(3,5-dimethylphenyl)methyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,9aR)-3-(4-aminobutyl)-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(6-methylpyridazin-3-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-(2-methoxyethyl)pyrrolidin-2-one
2-(8-methoxy-4-methylquinolin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
3-{4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
N-ethyl-3-(2-fluorophenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
(2R,6R)-4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(1-methyl-1H-1,2,3-benzotriazol-5-yl)oxan-4-yl]acetamide
(4-{[1-(thiophene-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
4-(2,4-dioxoimidazolidin-1-yl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
1-{4-[2-(4-fluorophenyl)morpholine-4-carbonyl]phenyl}pyrrolidin-2-one
1-[(4aR,8aS)-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-decahydro-1,6-naphthyridin-6-yl]-2-phenylethan-1-one
3-methyl-7-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one