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N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
5-(4-fluorophenyl)-2-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-2H-1,2,3,4-tetrazole
5-(3-methoxyphenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-pyrazole-3-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(pyrrolidin-1-yl)ethyl]amine
N-cyclopropyl-2-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
6-tert-butyl-1-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(4H-1,2,4-triazol-3-yl)piperidine
(3S,4S)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[ethyl(methyl)amino]-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(4aS,8aR)-6-(1,3-dihydroxypropan-2-yl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
methyl 2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-2-phenylacetate
4-(5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}pyrimidin-2-yl)morpholine
(3S,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-{3-[3-(6-methoxypyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(morpholin-4-yl)propanamide
1-(3-{[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indol-1-yl)ethan-1-one
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-cyclopentyl-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(carbamoylamino)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
3-(phenoxymethyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
N-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
3-[(3R,4S)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-(4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
N-methyl-2-(3-methylphenoxy)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
N,2-dimethyl-N-{1-[1-(pyridin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}benzamide
2-(pyridin-3-yl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-{2-[3-(1H-pyrazol-1-yl)propyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
4-hydroxy-N-[2-(pyridin-2-ylsulfanyl)ethyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
7-(5-chloropyridin-2-yl)-4-(5-methylpyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[(3S,5R)-1-benzyl-5-(piperidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
4-ethyl-1-[2-(1H-indol-3-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-oxopyrrolidin-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]-N-(propan-2-yl)benzamide
N-[(3,4-difluorophenyl)methyl]-1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-amine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-chloro-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-methyl-1H-pyrazole
N-{4-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]phenyl}acetamide
5-(4,4-difluoropiperidin-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-methyl-N-[4-methyl-3-({[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)phenyl]butanamide
4-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-methyl-1H-1,2,4-triazol-5-yl}morpholine
1-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(2-methylphenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
3-({4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
8-(5-chloropyridine-2-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2-cyclopentyl-N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
(3S,4S)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-methylpiperidine-3,4-diol