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(2S)-3-phenyl-2-[2-(2,3,6-trimethylphenoxy)acetamido]propanamide
1-(4-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}thiophen-2-yl)ethan-1-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(pyridin-4-ylmethyl)piperidin-4-ol
(3R,4R)-1-(5-fluoro-3,8-dimethylquinolin-2-yl)-4-(hydroxymethyl)piperidin-3-ol
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
5-(5-{[(4-methylphenyl)sulfanyl]methyl}furan-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-(1-benzofuran-2-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-[1-(cyclohexylmethyl)piperidin-4-yl]-N-cyclopropylpropanamide
1-[1-(2-hydroxyacetyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-(6-methylpyridazin-3-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}methanesulfonamide
N-{[7-(2-phenoxyacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
2-[(4aR,7aS)-4-(2-methyl-1H-pyrrole-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,4R)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
3-(4-cyclohexylpiperazine-1-carbonyl)-6-(2,5-dimethoxyphenyl)-N,N-dimethylpyridin-2-amine
(cyclohex-3-en-1-ylmethyl)[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(pyridin-3-yl)piperazin-1-yl]ethan-1-one
3-cyclopropyl-5-[2-(3,4-dimethyl-1H-pyrazol-5-yl)ethyl]-1,2,4-oxadiazole
N-[2-(1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]acetamide
(1R,3s,6r,8S)-4-[3-(piperidin-4-ylmethyl)benzoyl]-4-azatricyclo[4.3.1.13,8]undecane
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-aminopyrimidin-5-yl)-5,7-dimethyl-N-(1,1,1-trifluoropropan-2-yl)quinoline-4-carboxamide
5-chloro-2-(2-chloro-6-methoxyphenyl)pyrimidine
8-[(2R)-2-aminopropanoyl]-3-{2-[methyl(2-phenylethyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-ethyl-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(pyridin-4-ylmethyl)pentanamide
dimethyl(3-{2-[1-(3-methylpyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(3R,5S)-5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyrrolidin-3-amine
1-[4-(ethylsulfanyl)phenyl]-3-(2,2,2-trifluoroethyl)urea
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-phenylpyridine-3-carboxylic acid
4-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}thiomorpholine
N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)thiophene-2-sulfonamide
8-[(5-acetylthiophen-3-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
6-[2-(2-aminoethyl)morpholin-4-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
methyl 3-(furan-3-amido)-5-[(1-methoxypropan-2-yl)amino]-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-methyl-3-phenyl-1-(1,3,4-thiadiazol-2-yl)piperidine
2-(5-fluoro-2-methoxyphenyl)-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetic acid
2-(4-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenoxy)ethan-1-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
7-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(4aS,7aR)-N-(2,4-dimethylphenyl)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[3-(piperidine-1-carbonyl)phenyl]urea
ethyl 2-({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate