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4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-methoxyquinoline
2-ethyl-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-hydroxy-4-methyl-1-[4-(2-methylphenoxy)piperidin-1-yl]pentan-1-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amine
N-ethyl-2,8-dimethyl-N-[2-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
5-methoxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-oxo-1,4-dihydropyridine-2-carboxamide
3-[2-(1H-imidazol-4-yl)ethyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-{3-[({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenyl}ethan-1-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(quinolin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
[3-(cyclopropylmethyl)-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperidin-3-yl]methanol
1-(3-chloro-4-fluorophenyl)-4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazine
1-(1-{[3-(4-chlorophenoxy)phenyl]methyl}piperidin-4-yl)-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-(2-methylpropyl)pyrimidin-2-amine
2-({methyl[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(4-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(dimethylamino)ethan-1-one
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-4-phenyl-1H-imidazole-5-carboxamide
4-ethyl-3-{1-[3-(pyrimidin-2-yloxy)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-2-one
2-benzyl-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]acetamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetic acid
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-4,4,4-trifluorobutan-1-one
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-methyl-4-{[(2R,5S)-5-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}oxolan-2-yl]methyl}piperazine
(1S,5R)-6-(cyclobutylmethyl)-3-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(oxan-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{[(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyrimidine
4-({3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}methyl)pyridine
{2-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,3-thiazol-4-yl}methanol
N-ethyl-2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyridine-4-carboxamide
N-[2-({1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]pyridine-3-carboxamide
2-amino-1-{4-[4-({methyl[(1S)-1-phenylethyl]amino}methyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-4-(oxolan-2-ylmethyl)piperazine-1-carboxamide
4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-N-cyclopropylpiperazine-2-carboxamide
(3aS,6aS)-1-oxo-2-propyl-5-{thieno[3,2-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-(pyridin-2-ylmethyl)-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
N-[(3-phenoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-(naphthalen-2-yl)ethan-1-one
4-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]phenyl}-2-methylbutan-2-ol