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N-methyl-5-oxo-1-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrrolidine-3-carboxamide
1-methyl-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(1,3,4-thiadiazol-2-yl)urea
3-(2-chloro-5-sulfamoylphenyl)-1-[1-(cyclohex-1-en-1-yl)ethyl]urea
[(2,5-dimethoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
(1S,6R)-9-[2-(4-methylbenzoyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
[1-(5-fluoro-4-methoxypyrimidin-2-yl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
2-(furan-2-yl)-1-[2-(morpholin-4-yl)benzoyl]azepane
N-[2-methoxy-5-({[4-(oxolan-2-yl)butyl]carbamoyl}amino)phenyl]acetamide
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)pent-4-enamide
1-methyl-4-({5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
2,3-dimethyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]quinoxaline-6-carboxamide
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]morpholine-2-carboxylic acid
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-benzyl-3-ethyl-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-5-one
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperazine-1-sulfonamide
2-amino-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[2-(benzylsulfanyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(4-amino-3-hydroxybutanoyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S,4S)-1-methyl-4-[4-(thiophen-2-yl)butanamido]pyrrolidine-2-carboxylate
2-{1,4-bis[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
6-[(diethylamino)methyl]-N-(1-phenylcyclopropyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-hydroxy-1-(thian-4-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
2-({[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}amino)pyridine-4-carboxamide
1-cyclopentanecarbonyl-N-[3-(pyridin-4-yl)propyl]piperidine-4-carboxamide
1-({2-[3-(dimethylamino)-2-hydroxypropoxy]-5-methoxyphenyl}methyl)azetidin-3-ol
(1S,2S)-2-[4-(2,3-dimethylquinoxaline-6-carbonyl)piperazin-1-yl]cyclohexan-1-ol
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
N-[4-({2-[(2-chlorophenyl)methyl]morpholin-4-yl}methyl)phenyl]acetamide
N-[2-(4-fluorophenyl)ethyl]-1-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3,3,3-trifluoropropan-1-one
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(3-fluorophenyl)-4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)piperazin-2-one
(2S,4R)-4-amino-1-[5-(4-methoxyphenyl)furan-2-carbonyl]-N-methylpyrrolidine-2-carboxamide
N-(6-methoxyquinolin-8-yl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
N-[(2R,4R,6S)-2-tert-butyl-6-[2-(methoxymethyl)pyrimidin-5-yl]oxan-4-yl]acetamide
N-[4-(azepan-1-yl)butyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
3,5-dimethoxy-2-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzoic acid
1-ethyl-5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-(propan-2-yl)-1H-pyrazole
7-[4-(trifluoromethyl)benzoyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
(2S,4R)-4-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamido]-N-(propan-2-yl)-1-propylpyrrolidine-2-carboxamide
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-methylpropyl)-6-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,6-dihydropyridine-3-carboxamide