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N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4-methoxybenzamide
(3S,9aR)-8-[(2-fluorophenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
N-[4-(pyridin-3-yloxy)phenyl]-1-(1,3-thiazol-4-ylmethyl)piperidine-2-carboxamide
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-1-benzofuran-5-carboxamide
1-(2,6-difluoro-3-methoxybenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-amino-4-ethyl-6-(2-fluorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(azepan-1-yl)-4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]butane-1,4-dione
1-[4-({[2-(4-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(diethylamino)propan-2-ol
6-{3-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
(2S)-2-amino-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
N-[(4-fluorophenyl)methyl]-6-oxo-N-(1-phenylethyl)-1,6-dihydropyridazine-3-carboxamide
5-ethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]pyrimidin-2-amine
5-[(3-methoxypiperidin-1-yl)methyl]-2-(propan-2-yl)pyrimidine
2-methoxy-1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
2-(3-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[(3-methylpyridin-4-yl)methyl]piperidine-4-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide
N-cyclopentyl-1-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}morpholine
3-{[1-butyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,2-oxazinane
3-(2,5-dimethoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
4-{5-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-4-fluorobenzamide
(2-{2-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
[1-(2-fluorophenyl)propan-2-yl]({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
4-hydroxy-1-[2-(1H-pyrazol-1-yl)butanoyl]piperidine-4-carboxylic acid
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[2-hydroxy-2-(thiophen-2-yl)ethyl]urea
4-[1-(3-methylbutyl)-5-(5-phenoxyfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-{4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1-methylpiperazin-2-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
3-(3-methoxypropyl)-1-[2-(2H-1,2,3-triazol-2-yl)acetyl]piperidine-3-carboxylic acid
1-(2-fluorophenyl)-2,2-dimethyl-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]cyclopropane-1-carboxamide
(5-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}furan-2-yl)methanol
1-(4-methylpentanoyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
5-ethyl-N,2-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
4-chloro-N-{2-[4-(dimethyl-1,2-oxazol-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethoxybenzamide
3-[2-(4-fluorophenyl)ethyl]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[(2,3-dichloro-6-fluorophenyl)methyl]-3-methylimidazolidin-2-one
4-(azepane-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-cyclobutanecarbonyl-1'-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(3-acetylphenoxymethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
2-ethyl-4-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyrimidine
1,3-dimethyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
6-methyl-2-({2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
N-[2-(dimethylamino)ethyl]-5-(3-methylpyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide