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N-[(1-cyclobutanecarbonylpiperidin-3-yl)methyl]-4-fluorobenzamide
4-(4-fluoro-2-methylphenoxy)-1-(furan-3-ylmethyl)piperidine-4-carboxylic acid
N-[(3-chlorophenyl)methyl]-5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
3-[3-(dimethylamino)propyl]-1-[4-(3-methoxyphenoxy)phenyl]-3-methylurea
3-[(4-ethylpiperazin-1-yl)methyl]-7-fluoro-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydroquinolin-2-one
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
2-(2-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}phenoxy)acetic acid
3-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-[(2-chlorophenyl)methyl]propanamide
(1R,3S)-3-amino-N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-4-ylmethyl)cyclohexane-1-carboxamide
1-(pyrazin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
N4-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
(2R,3R,6R)-5-(4-methoxybenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(1-methyl-1H-pyrazol-5-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(2S,4R)-4-[2-(4-chlorophenyl)acetamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N,N-dimethylacetamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-(3-chlorophenyl)-4-[3-(thiophen-3-yl)propanoyl]piperazin-2-one
1-{5-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2-methyl-1,3-benzothiazole
N-[2-(2-chlorophenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)spiro[2.4]heptane-1-carboxamide
2-cyclopropanecarbonyl-8-{furo[3,2-c]pyridin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,3,4,7-tetramethyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
2-(5-fluoro-2-methylphenyl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
3-{2-[2-(benzyloxy)phenyl]-1H-imidazol-1-yl}propan-1-ol
3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-1-{2-[(pyridin-3-yl)amino]ethyl}urea
(1S,5R)-N-(3-methylphenyl)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(5-chloropyridin-2-yl)acetamide
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
[(1S,3S,3aS,6aR)-5-methyl-1-phenyl-3-(1-phenyl-1H-pyrazol-4-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-N-[2-(3-chlorophenoxy)ethyl]-3-ethyl-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[4-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
6-(3-fluorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N4-ethyl-N2-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-2,4-diamine
2-[(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
2-(4-tert-butylphenyl)-2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}acetic acid
1-[1-methyl-4-(oxolan-3-ylmethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]-3-phenylpropan-1-one
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-cyclopentyl-5-[(8-methoxyquinolin-2-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1,5-dimethyl-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-(2-chlorophenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}furan-2-carboxamide
3-[(2,2-dimethylmorpholin-4-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-{1'-[2-(morpholin-3-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-imidazole-2-carboxamide
1-amino-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}cyclopropane-1-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]methanol