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benzyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(prop-2-yn-1-yl)amine
1-(2-fluorophenyl)-4-[(4-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
N-[2-(ethylsulfanyl)ethyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
6-cyano-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-3-carboxamide
4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]pyridine-2-carboxylic acid
N,8-dimethyl-3-{[(oxan-2-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-{[1-(hydroxymethyl)cyclopentyl]methyl}-1-[3-(3-methoxyphenyl)phenyl]-3-methylurea
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
2-methyl-7-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-methyl-4-{5-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}piperidine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(thiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-fluoro-3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)benzene-1-sulfonamide
2-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-9-oxa-2-azaspiro[5.5]undecane
1-[2-(4-chlorophenyl)ethyl]-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
2-[8-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
N-(1,3-dihydroxypropan-2-yl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
6-methoxy-2-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-{[2-(5-methoxypyridin-3-yl)phenyl]methyl}propanamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-methyl-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(2-methoxyethyl)-2-(5-phenyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
6-ethoxy-2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}quinoline
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-2-(3-methoxypiperidin-1-yl)pyrimidine
1-cyclopentyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-6-oxopiperidine-3-carboxamide
ethyl 4-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}amino)piperidine-1-carboxylate
2-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(1H-1,2,3-benzotriazol-4-yl)-3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methylurea
2-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine-3-carbonyl)pyridine
2-{[4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)phenyl](methyl)amino}ethan-1-ol
3-{3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
N-(cyclohexylmethyl)-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
3-[1-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]adamantan-1-ol
1-{4-[4-(1H-pyrazol-1-yl)phenyl]phenyl}propan-1-ol
(3R,4S)-1-[5-(methanesulfonylmethyl)pyridin-2-yl]-4-propylpyrrolidin-3-amine
5-{3-[3-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}(3-phenylpropyl)amine
5-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-2-methyl-1,3-benzothiazole
2-oxo-N-[1-(thian-4-yl)piperidin-4-yl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(2-methoxyethyl)-1-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
4-{6-[3-(benzyloxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
{1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-4-yl}methanol
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
(2S,4S)-4-amino-1-(1-methyl-1H-indazole-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{1-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-1-oxopropan-2-yl}methanesulfonamide
N-[2-(N-methylmethanesulfonamido)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-(4-fluorophenyl)-N-(2-methylpropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-{4-[1-(methylamino)propyl]phenyl}benzamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine