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dimethyl(3-{2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}but-3-en-1-one
N-{2-[(4-fluorophenyl)formamido]ethyl}-3-(1,2-oxazinan-2-yl)propanamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-3-[(3-methylpiperidin-1-yl)methyl]benzamide
8-(3-aminothiophene-2-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]thiophene-2-carboxamide
4-[({3-[(dimethylamino)methyl]phenyl}methyl)amino]pyrimidine-5-carboxylic acid
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-(furan-2-ylmethyl)-3-(2-hydroxyethyl)urea
N-methyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-N-(2-phenylethyl)piperidin-3-amine
6-methoxy-3-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-benzofuran-2-carboxamide
3-hydroxy-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
[(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-(prop-2-en-1-yl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidine-3-carboxylic acid
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-({7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
2-(4-{[cyclopentyl(prop-2-en-1-yl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
7-(2-methoxyethyl)-2-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
2-(2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3,4-dimethoxybenzoyl)piperidine
1-benzyl-N-ethyl-4-oxo-5-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
3-(oxan-4-yl)-5-(oxolan-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
N-(3-fluorophenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-amine
N-(4-fluoro-2-methylphenyl)-3-[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]propanamide
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(pyridin-3-yl)acetamide
1-(1-ethylpiperidine-2-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N,N-dimethyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(1,4-dithiepan-6-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(4-{[6-(4-methoxyphenyl)-7-oxo-6,9-diazaspiro[4.5]decan-9-yl]methyl}phenyl)acetamide
5-propyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,2-oxazole-3-carboxamide
N-cyclobutyl-4-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]morpholine-2-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}cyclopropanamine
N-(2-methylpropyl)-1-[1-(pentan-3-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
7-(cyclobutylmethyl)-2-[(2,4,5-trimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(piperidine-1-carbonyl)piperidine
2-(4-methoxyphenyl)-N-({1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methyl)acetamide
N,6-dimethyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}pyridine-2-carboxamide
(2S,4R)-4-amino-N-methyl-1-(4-phenoxybutanoyl)pyrrolidine-2-carboxamide
3-amino-N-[3-(cyclopentyloxy)phenyl]pyrrolidine-1-carboxamide
3-phenyl-1-{1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl}propan-1-one
4-(5-acetylpyridin-2-yl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-fluorobutyl)-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methoxyquinoline
2-(1-methyl-1H-pyrazole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
2-({3-azaspiro[5.5]undecan-9-yl}amino)-N-(5-fluoro-2-methylphenyl)propanamide