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4-(3-ethyl-1H-pyrazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(pyridin-4-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
N-[(2S,4R,6S)-2-benzyl-6-[(benzyloxy)methyl]oxan-4-yl]acetamide
2-[N-(3-fluorophenyl)methanesulfonamido]-N-(1-hydroxypropan-2-yl)acetamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
(1S,5R)-6-benzyl-3-[2-oxo-2-(piperazin-1-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylthian-4-amine
2-{[4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenol
1-cyclohexyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-6-[2-(3-methylbut-2-en-1-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
[(5-chlorofuran-2-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
(5-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}furan-2-yl)methanol
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2,2-dimethyloxan-4-yl)benzamide
(1S,5R)-6-(2-methoxyethyl)-3-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2-ethoxyphenyl)methyl]piperidine
N-methyl-2-(5-methyl-3-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carbonyl}-1H-pyrazol-1-yl)acetamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
5-methoxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-2-amine
5-(azepan-1-yl)-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(furan-2-ylmethyl)-N-methylbenzamide
methyl 4-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazine-1-carboxylate
5-{4-[1-(dimethylamino)ethyl]piperidine-1-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
2-cyclobutyl-9-(2-phenylpropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetyl}-3,3-dimethylpiperazin-2-one
5-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-2-methoxyphenol
(4aS,7aR)-1-(2-ethylpyrimidine-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1,3-dimethyl-N-[(2,3,4,5-tetrafluorophenyl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoxalin-2-ol
N-[3-hydroxy-1-(4-methylphenyl)propyl]-3-(1-methylpiperidin-4-yl)propanamide
2-(4-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}morpholin-3-yl)-1-(pyrrolidin-1-yl)ethan-1-one
methyl 2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-3-carboxylate
(2S,4R)-4-amino-1-(5-methyl-4-phenylthiophene-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-ethyl-1-methyl-3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-ethyl-5-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
5-acetyl-2,4-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-1H-pyrrole-3-carboxamide
(1S,5R)-6-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-4-[2-(4-fluorophenoxy)ethyl]-1,4-diazepan-5-one
3-{2-[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
(2S,4R)-1-(1H-imidazol-2-ylmethyl)-N-(propan-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
3-[(ethylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-butyl-5-(2-methoxypyridin-3-yl)furan-2-carboxamide
5-methoxy-4-oxo-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1,4-dihydropyridine-2-carboxamide
5-methoxy-2-[5-(prop-2-ene-1-sulfonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
N-[3-(dimethylcarbamoyl)phenyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide